SB-277011 hydrochloride
Cat. No. :YN320363
CAS No. :215804-67-4
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order@ubiochem.com| Product Name: | SB-277011 hydrochloride |
| CAS NO.: | 215804-67-4 |
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| Molecular Weight: | 475.02 |
| Molecular Formula: | C₂₈H₃₁ClN₄O |
| SMILES: | O=C(C1=CC=NC2=CC=CC=C21)N[C@@H]3CC[C@H](CC3)CCN4CC5=C(CC4)C=C(C#N)C=C5.[H]Cl |
| Storage: | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Transportation: | Room temperature in continental US; may vary elsewhere. |
| Description: | SB-277011 hydrochloride (SB-277011A hydrochloride) is a potent, selective, orally bioavailable and brain penetratedopamine D3receptor (D3R)antagonist with Ki values of 10.7 nM and 11.2nM at rodent and human D3R, respectively. SB-277011 hydrochloride displays 80- to 100-fold selectivity over other dopamine receptors withpKis of 8.0, 6.0, <5.2, and 5.9 for D3, D2, 5-HT1B, and 5-HT1Dreceptors, respectively. |
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