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Cannabinoid Receptor

Chemical structure

Cat.No.

Product Name

CAS no.

Target

  • YN321738 β-Caryophyllene 87-44-5

    β-Caryophyllene is a natural bicyclic sesquiterpene that is a constituent of many essential oils. It acts as a non-steroidal anti-inflammatory drug, a fragrance and a metabolite.

  • YN321395 Pregnenolone 145-13-1

    Pregnenolone is an endogenous steroid hormone, used in the treatment of fatigue, Alzheimer’s disease, trauma and injuries.

  • YN321736 Yangonin 500-62-9

    Yangonin is a novel CB₁ receptor ligand, it exhibits affinity for the human recombinant CB₁ receptor. Yangonin could be a valuable candidate for the intervention of NF-κB-dependent pathological conditions such as inflammation. ...

  • YN322097 Olivetol 500-66-3

    Olivetol is a naturally occurring organic compound being a precursor in various syntheses of tetrahydrocannabinol. It acts as a competitive inhibitor of the cannabinoid receptors CB1 and CB2.

  • YN321677 Pregnenolone monosulfate 1247-64-9

    Pregnenolone monosulfate (3β-Hydroxy-5-pregnen-20-one monosulfate) is a powerful neurosteroid, the main precursor of various steroid hormones including steroid ketones. Pregnenolone monosulfate acts as a signaling-specific inhibitor ofc...

  • YN320411 Pregnenolone monosulfate sodi... 1852-38-6

    Pregnenolone monosulfate sodium salt (3β-Hydroxy-5-pregnen-20-one monosulfate sodium salt) is a powerful neurosteroid, the main precursor of various steroid hormones including steroid ketones. Pregnenolone monosulfate sodium salt acts a...

  • YN320466 N-Oleoyl glycine 2601-90-3

    N-Oleoyl glycine is a lipoamino acid, which stimulates adipogenesis associated with activation ofCB1 receptor and Aktsignaling pathway in 3T3-L1 adipocyte.

  • YN320984 BML-190 2854-32-2

    BML-190(IMMA) is a potent and selective CB2 receptor lig and (Ki values are 435nM and > 2μM for CB2 and CB1 respectively).

  • YN321770 Voacamine 3371-85-5

    Voacamine, an indole alkaloid, isolated fromVoacanga Africana, exhibits potentcannabinoid CB1 receptorantagonistic activity. Voacamine also inhibitsP-glycoprotein(P-gp) action in multidrug-resistant tumor cells.

  • YN320408 Leelamine hydrochloride 16496-99-4

    Leelamine hydrochloride is a tricyclic diterpene molecule that is extracted from the bark of pine trees. Leelamine hydrochloride is acannabinoid receptor type 1 (CB1)agonist and a inhibitor of SREBP1-regulatedfatty acid/lipid syn...

  • YN320502 Tetrahydromagnolol 20601-85-8

    Tetrahydromagnolol (Magnolignan), a main metabolite of Magnolol, is a potent and selectivecannabinoid CB2 receptoragonist with an EC50 of 170nM and a Ki of 416nM. Tetrahydromagnolol possesses 20-fold more selective forCB2 r...

  • YN322106 2-Palmitoylglycerol 23470-00-0

    2-Palmitoylglycerol (2-Palm-Gl), an congener of 2-arachidonoylglycerol (2-AG), is a modestcannabinoid receptor CB1agonist. 2-Palmitoylglycerol also may be an endogenous lig and for GPR119.

  • YN322103 2-Arachidonoylglycerol 53847-30-6

    2-Arachidonoylglycerol is a second endogenous cannabinoid lig and in the central nervous system.

  • YN320375 Anandamide 94421-68-8

    An and amide is an immune modulator in the central nervous system acts via not onlycannabinoid receptors(CB1 and CB2) but also other targets (e.g.,GPR18/GPR55).

  • YN320716 WIN 55,212-2 Mesylate 131543-23-2

    WIN 55,212-2 Mesylate is a potent aminoalkylindolecannabinoid (CB) receptoragonist with Kis of 62.3 and 3.3nM for human recombinant CB1 and CB2 receptors, respectively.

  • YN320985 6-Iodopravadoline 164178-33-0

    6-Iodopravadoline (AM630) is a selective cannabinoid CB2 receptor antagonist with Ki of 31.2 nM.

  • YN320821 Rimonabant 168273-06-1

    Rimonabant is a selective antagonist of CB1 with IC50 of 13.6 nM and EC50 of 17.3 nM in hCB1 transfected HEK 293 membrane.

  • YN320988 AM251 183232-66-8

    AM251 block the inhibitory effects of endocannabinoids and synthetic cannabinoid agonists on transmitter release through an action at presynaptic cannabinoid 1 receptors in brain.

  • YN320735 SR144528 192703-06-3

    SR144528 is a potent and selectiveCB2 receptorantagonist with a Ki of 0.6nM.

  • YN320740 AM281 202463-68-1

    AM281 is a selectiveCB1 receptorantagonist with an IC50 of 9.91nM. AM281 inhibits CB2 receptor with an IC50 of 13000nM.

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