β-Caryophyllene is a natural bicyclic sesquiterpene that is a constituent of many essential oils. It acts as a non-steroidal anti-inflammatory drug, a fragrance and a metabolite.
Pregnenolone is an endogenous steroid hormone, used in the treatment of fatigue, Alzheimer’s disease, trauma and injuries.
Yangonin is a novel CB₁ receptor ligand, it exhibits affinity for the human recombinant CB₁ receptor.
Yangonin could be a valuable candidate for the intervention of NF-κB-dependent pathological conditions such as inflammation.
Olivetol is a naturally occurring organic compound being a precursor in various syntheses of tetrahydrocannabinol. It acts as a competitive inhibitor of the cannabinoid receptors CB1 and CB2.
Pregnenolone monosulfate (3β-Hydroxy-5-pregnen-20-one monosulfate) is a powerful neurosteroid, the main precursor of various steroid hormones including steroid ketones. Pregnenolone monosulfate acts as a signaling-specific inhibitor ofc...
Pregnenolone monosulfate sodi...
Pregnenolone monosulfate sodium salt (3β-Hydroxy-5-pregnen-20-one monosulfate sodium salt) is a powerful neurosteroid, the main precursor of various steroid hormones including steroid ketones. Pregnenolone monosulfate sodium salt acts a...
N-Oleoyl glycine is a lipoamino acid, which stimulates adipogenesis associated with activation ofCB1 receptor and Aktsignaling pathway in 3T3-L1 adipocyte.
BML-190(IMMA) is a potent and selective CB2 receptor lig and (Ki values are 435nM and > 2μM for CB2 and CB1 respectively).
Voacamine, an indole alkaloid, isolated fromVoacanga Africana, exhibits potentcannabinoid CB1 receptorantagonistic activity. Voacamine also inhibitsP-glycoprotein(P-gp) action in multidrug-resistant tumor cells.
Leelamine hydrochloride is a tricyclic diterpene molecule that is extracted from the bark of pine trees. Leelamine hydrochloride is acannabinoid receptor type 1 (CB1)agonist and a inhibitor of SREBP1-regulatedfatty acid/lipid syn...
Tetrahydromagnolol (Magnolignan), a main metabolite of Magnolol, is a potent and selectivecannabinoid CB2 receptoragonist with an EC50 of 170nM and a Ki of 416nM. Tetrahydromagnolol possesses 20-fold more selective forCB2 r...
2-Palmitoylglycerol (2-Palm-Gl), an congener of 2-arachidonoylglycerol (2-AG), is a modestcannabinoid receptor CB1agonist. 2-Palmitoylglycerol also may be an endogenous lig and for GPR119.
An and amide is an immune modulator in the central nervous system acts via not onlycannabinoid receptors(CB1 and CB2) but also other targets (e.g.,GPR18/GPR55).
WIN 55,212-2 Mesylate
WIN 55,212-2 Mesylate is a potent aminoalkylindolecannabinoid (CB) receptoragonist with Kis of 62.3 and 3.3nM for human recombinant CB1 and CB2 receptors, respectively.
Rimonabant is a selective antagonist of CB1 with IC50 of 13.6 nM and EC50 of 17.3 nM in hCB1 transfected HEK 293 membrane.
AM251 block the inhibitory effects of endocannabinoids and synthetic cannabinoid agonists on transmitter release through an action at presynaptic cannabinoid 1 receptors in brain.
AM281 is a selectiveCB1 receptorantagonist with an IC50 of 9.91nM. AM281 inhibits CB2 receptor with an IC50 of 13000nM.
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