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DYRK

Chemical structure

Cat.No.

Product Name

CAS no.

Target

  • YN440349 ID-8 147591-46-6

    ID-8 is a DYRK inhibitor, and sustains embryonic stem cell self-renewal in long-term culture.

  • YN440271 LDN-192960 184582-62-5

    LDN-192960 is an inhibitor ofHaspin and Dual-specificity Tyrosine-regulated Kinase 2 (DYRK2)with IC50s of 10nM and 48nM, respectively.

  • YN440105 GSK-626616 1025821-33-3

    GSK-626616 is a potent, orally bioavailable inhibitor ofDYRK3(IC50=0.7nM). GSK-626616 inhibits other members of the DYRK family (e.g., DYRK1A and DYRK2) with similar potency, which is a potential therapy for the ...

  • YN440112 INDY 1169755-45-6

    INDY is a potent and ATP-competitiveDyrk1A and Dyrk1Binhibitor with IC50s of 0.24μM and 0.23μM, respectively. INDY binds in the ATP pocket of the enzyme and has aKivalue of 0.18μM for Dyrk1A. INDY shar...

  • YN440448 Protein kinase inhibitors 1 1365986-44-2

    Protein kinase inhibitors 1 is a novel inhibitor ofHIPK2with an IC50 of 74nM and Kdof 9.5nM.

  • YN440225 Mirk-IN-1 1386979-55-0

    Mirk-IN-1 is a potent inhibitor of Dyrk1B(Mirk kianse) and Dyrk1A with IC50 of 68±48nM and 22±8nM respectively.

  • YN440199 AZ191 1594092-37-1

    AZ191 is a potent and selective DYRK1B inhibitor with IC50 of 17 nM in a cell-free assay, about 5- and 110-fold selectivity over DYRK1A and DYRK2, respectively.

  • YN440013 tBID 1639895-85-4

    tBID is a selective inhibitor of homeodomain-interacting protein kinase 2 (HIPK2) with an IC50 of  0.33 µM.

  • YN440173 AZ-Dyrk1B-33 1679330-37-0

    AZ-Dyrk1B-33 is a potent and selectiveDyrk1B kinaseinhibitor, with an IC50 of 7nM.

  • YN440169 CLK-IN-T3 2109805-56-1

    CLK-IN-T3 is a high potent, selective, and stableCDC-like kinase (CLK)inhibitor with IC50s of 0.67nM, 15nM, and 110nM for CLK1, CLK2, and CLK3 protein kinases, respectively. CLK-IN-T3 has anti-cancer ac...

  • YN440272 LDN-192960 hydrochloride 2309172-48-1

    LDN-192960 hydrochloride is an inhibitor ofHaspin and Dual-specificity Tyrosine-regulated Kinase 2 (DYRK2)with IC50s of 10nM and 48nM, respectively.

  • YN440199 AZ191

    AZ191 is a potent and selective DYRK1B inhibitor with IC50 of 17 nM in a cell-free assay, about 5- and 110-fold selectivity over DYRK1A and DYRK2, respectively.

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