Chemical structure
Cat.No.
Product Name
CAS no.
Target
ID-8 is a DYRK inhibitor, and sustains embryonic stem cell self-renewal in long-term culture.
YN440271 LDN-192960 184582-62-5
LDN-192960 is an inhibitor ofHaspin and Dual-specificity Tyrosine-regulated Kinase 2 (DYRK2)with IC50s of 10nM and 48nM, respectively.
YN440105 GSK-626616 1025821-33-3
GSK-626616 is a potent, orally bioavailable inhibitor ofDYRK3(IC50=0.7nM). GSK-626616 inhibits other members of the DYRK family (e.g., DYRK1A and DYRK2) with similar potency, which is a potential therapy for the ...
INDY is a potent and ATP-competitiveDyrk1A and Dyrk1Binhibitor with IC50s of 0.24μM and 0.23μM, respectively. INDY binds in the ATP pocket of the enzyme and has aKivalue of 0.18μM for Dyrk1A. INDY shar...
YN440448 Protein kinase inhibitors 1 1365986-44-2
Protein kinase inhibitors 1 is a novel inhibitor ofHIPK2with an IC50 of 74nM and Kdof 9.5nM.
YN440225 Mirk-IN-1 1386979-55-0
Mirk-IN-1 is a potent inhibitor of Dyrk1B(Mirk kianse) and Dyrk1A with IC50 of 68±48nM and 22±8nM respectively.
AZ191 is a potent and selective DYRK1B inhibitor with IC50 of 17 nM in a cell-free assay, about 5- and 110-fold selectivity over DYRK1A and DYRK2, respectively.
tBID is a selective inhibitor of homeodomain-interacting protein kinase 2 (HIPK2) with an IC50 of 0.33 µM.
YN440173 AZ-Dyrk1B-33 1679330-37-0
AZ-Dyrk1B-33 is a potent and selectiveDyrk1B kinaseinhibitor, with an IC50 of 7nM.
YN440169 CLK-IN-T3 2109805-56-1
CLK-IN-T3 is a high potent, selective, and stableCDC-like kinase (CLK)inhibitor with IC50s of 0.67nM, 15nM, and 110nM for CLK1, CLK2, and CLK3 protein kinases, respectively. CLK-IN-T3 has anti-cancer ac...
YN440272 LDN-192960 hydrochloride 2309172-48-1
LDN-192960 hydrochloride is an inhibitor ofHaspin and Dual-specificity Tyrosine-regulated Kinase 2 (DYRK2)with IC50s of 10nM and 48nM, respectively.
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