ULS |Focus on small molecule Inhibitors&Agonists

Inhibitors & Agonists
- Anti-infection
  - Antibiotic
  - Arenavirus
  - Bacterial
  - CMV
  - Enterovirus
  - Filovirus
  - Fungal
  - HBV
  - HCV
  - HCV Protease
  - HIV
  - HIV Protease
  - HSV
  - Influenza Virus
  - Parasite
  - ReverseTranscriptase
  - RSV
  - SARS-CoV
  - Virus Protease
  - Reverse Transcriptase
- ADC Related
  - ADC cytotoxin
  - ADC linker
  - Drug-Linker Conjugates for ADC
  - PROTAC-linker Conjugate for PA
- Apoptosis
  - Apoptosis
  - Bcl-2 Family
  - c-Myc
  - Caspase
  - DAPK
  - Ferroptosis
  - FKBP
  - IAP
  - MDM-2/p53
  - PKD
  - Pyroptosis
  - RIP kinase
  - Survivin
  - Thymidylate Synthase
  - TNF Receptor
- Autophagy
  - FKBP
  - LRRK2
  - Mitophagy
  - ULK
  - Autophagy
- Cell cycle/DNA damage
  - Antifolate
  - APC
  - ATM/ATR
  - Aurora Kinase
  - Casein Kinase
  - CDK
  - Checkpoint Kinase (Chk)
  - CRISPR/Cas9
  - Deubiquitinase
  - DNA Alkylator/Crosslinker
  - DNA-PK
  - DNA/RNA Synthesis
  - Eukaryotic Initiation Factor (
  - G-quadruplex
  - Haspin Kinase
  - HDAC
  - HSP
  - IRE1
  - Kinesin
  - LIM Kinase (LIMK)
  - Microtubule/Tubulin
  - Mps1
  - Nucleoside Antimetabolite/Anal
  - p97
  - PAK
  - PARP
  - PERK
  - Polo-like Kinase (PLK)
  - PPAR
  - RAD51
- Cytoskeleton
  - Arp2/3 Complex
  - Dynamin
  - Gap Junction Protein
  - Integrin
  - Kinesin
  - Microtubule/Tubulin
  - Mps1
  - Myosin
  - PAK
  - ROCK
- Epigenetics
  - AMPK
  - Aurora Kinase
  - DNA Methyltransferase
  - Epigenetic Reader Domain
  - HDAC
  - Histone Acetyltransferase
  - Histone Demethylase
  - Histone Methyltransferase
  - JAK
  - MicroRNA
  - PARP
  - PKC
  - Protein Arginine Deiminase
  - Sirtuin
- GPCR/G Protein
  - 5-HT Receptor
  - Adenosine Receptor
  - Adenylate Cyclase
  - Adiponectin Receptor
  - Adrenergic Receptor
  - Angiotensin Receptor
  - Bombesin Receptor
  - Bradykinin Receptor
  - Cannabinoid Receptor
  - CaSR
  - CCR
  - CGRP Receptor
  - Cholecystokinin Receptor
  - CRFR
  - CXCR
  - Dopamine Receptor
  - EBI2/GPR183
  - Endothelin Receptor
  - GHSR
  - Glucagon Receptor
  - Glucocorticoid Receptor
  - GNRH Receptor
  - GPCR19
  - GPR109A
  - GPR119
  - GPR120
  - GPR139
  - GPR40
  - GPR55
  - GPR84
- Immunology/Inflammation
  - Arginase
  - CCR
  - Aryl Hydrocarbon Receptor
  - CD73
  - Complement System
  - COX
  - CXCR
  - Cyclic GMP-AMP Synthase
  - FKBP
  - FLAP
  - Galectin
  - Histamine Receptor
  - IFNAR
  - Interleukin Related
  - IRAK
  - MyD88
  - NO Synthase
  - NOD-like Receptor (NLR)
  - PD-1/PD-L1
  - PGE synthase
  - Pyroptosis
  - Reactive Oxygen Species
  - Salt-inducible Kinase (SIK)
  - SPHK
  - STING
  - Thrombopoietin Receptor
  - Toll-like Receptor (TLR)
- JAK/STAT Signaling
  - EGFR
  - JAK
  - Pim
  - STAT
- MAPK/ERK Pathway
  - KLF
  - JNK
  - ERK
  - MAP3K
  - MAP4K
  - MAPKAPK2 (MK2)
  - MEK
  - Mixed Lineage Kinase
  - MNK
  - p38 MAPK
  - Raf
  - Ribosomal S6 Kinase (RSK)
- Membrane Transporter/Ion Chann
  - Calcium Channel
  - BCRP
  - ATP Synthase
  - CFTR
  - Chloride Channel
  - CRAC Channel
  - CRM1
  - EAAT2
  - GABA Receptor
  - GLUT
  - GlyT
  - HCN Channel
  - iGluR
  - Monoamine Transporter
  - Monocarboxylate Transporter
  - Na+/Ca2+ Exchanger
  - Na+/HCO3- Cotransporter
  - Na+/K+ ATPase
  - nAChR
  - NKCC
  - P-glycoprotein
  - P2X Receptor
  - Potassium Channel
  - Proton Pump
  - SGLT
  - Sodium Channel
  - TRP Channel
  - VDAC
  - URAT1
- Metabolic Enzyme/Protease
  - Acyltransferase
  - Acetyl-CoA Carboxylase
  - 5 alpha Reductase
  - 15-PGDH
  - Aldehyde Dehydrogenase (ALDH)
  - Aldose Reductase
  - Aminoacyl-tRNA Synthetase
  - Aminopeptidase
  - Angiotensin-converting Enzyme
  - Arginase
  - ATGL
  - ATP Citrate Lyase
  - Carbonic Anhydrase
  - Carboxypeptidase
  - Cathepsin
  - CETP
  - COMT
  - Cytochrome P450
  - Dihydroorotate Dehydrogenase
  - Dipeptidyl Peptidase
  - Drug Metabolite
  - E1/E2/E3 Enzyme
  - Elastase
  - Endogenous Metabolite
  - Enolase
  - Epoxide Hydrolase
  - FABP
  - Factor Xa
  - Farnesyl Transferase
  - Fatty Acid Synthase (FASN)
- Neuronal Signaling
  - Adrenergic Receptor
  - Adenosine Kinase
  - AChE
  - 5-HT Receptor
  - Amyloid-β
  - Beta-secretase
  - Calcium Channel
  - CaMK
  - Cannabinoid Receptor
  - CGRP Receptor
  - Cholecystokinin Receptor
  - COMT
  - Dopamine Receptor
  - Dopamine Transporter
  - FAAH
  - GABA Receptor
  - GlyT
  - GPR119
  - GPR139
  - GPR55
  - Histamine Receptor
  - iGluR
  - Imidazoline Receptor
  - mAChR
  - MCHR1 (GPR24)
  - Melanocortin Receptor
  - Melatonin Receptor
  - mGluR
  - Monoamine Oxidase
  - nAChR
- PI3K/Akt/mTOR
  - Akt
  - AMPK
  - PTEN
  - PIKfyve
  - PI4K
  - PI3K
  - PDK-1
  - mTOR
  - MELK
  - DNA-PK
  - GSK-3
  - ATM/ATR
- NF-κB
  - IKK
  - Keap1-Nrf2
  - MALT1
  - NF-κB
  - Reactive Oxygen Species
- PROTAC
  - E3 Ligase Ligand-Linker Conjug
  - Ligand for E3 Ligase
  - Ligand for Target Protein for
  - PROTAC
  - PROTAC Linker
  - PROTAC-linker Conjugate for PA
  - SNIPER
  - Target Protein Ligand-Linker C
  - E3 Ligase Ligand-Linker Conjug
  - Ligand for Target Protein for
  - PROTAC-linker Conjugate for PA
  - Target Protein Ligand-Linker C
- Protein Tyrosine Kinase/RTK
  - Bcr-Abl
  - Ack1
  - ALK
  - Btk
  - c-Fms
  - c-Kit
  - c-Met/HGFR
  - Discoidin Domain Receptor
  - DYRK
  - EGFR
  - Ephrin Receptor
  - FAK
  - FGFR
  - FLT3
  - IGF-1R
  - Insulin Receptor
  - Itk
  - PDGFR
  - PKA
  - Pyk2
  - RET
  - ROS
  - Src
  - Syk
  - TAM Receptor
  - Trk Receptor
  - VEGFR
  - BMX Kinase
- Stem Cell/Wnt
  - Casein kinase
  - Gli
  - ERK
  - GSK-3
  - Hedgehog
  - Hippo (MST)
  - JAK
  - Notch
  - Oct3/4
  - PKA
  - Porcupine
  - ROCK
  - sFRP-1
  - Smo
  - STAT
  - TGF-beta/Smad
  - Wnt
  - YAP
  - β-catenin
  - γ-secretase
- TGF-beta/Smad
  - TGF-beta/Smad
  - ROCK
  - PKC
  - TGF-β Receptor
- Vitamin D related
  - VD / VDR
- Others
  - Androgen Receptor
  - Aromatase
  - Estrogen Receptor/ERR
  - Progesterone Receptor
  - Thyroid Hormone Receptor
  - Others
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