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CaSR

Chemical structure

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CAS no.

Target

  • YN321129 Strontium Ranelate 135459-87-9

    Strontium Ranelate (S12911) is an antiosteoporotic agent that acts by reducing bone resorption and promoting bone formation, thereby inducing a positive bone balance. Strontium Ranelate also can activate thecalcium-sensing receptor (...

  • YN320175 Tecalcet Hydrochloride 177172-49-5

    Tecalcet Hydrochloride (R 568 Hydrochloride), an orally active calcimimetic compound, allosterically and positively modulates thecalcium-sensing receptor (CaSR). Tecalcet Hydrochloride (R 568 Hydrochloride) increases the sensit...

  • YN321292 Cinacalcet 226256-56-0

    Cinacalcet (AMG073, Sensipar, Cin) is an orally active, allosteric agonist of receptors for calcium (CaR) that increases the sensitivity of the CaR to Ca.

  • YN321722 Ligustroflavone 260413-62-5

    Ligustroflavone, isolated from the leaves of Turpinia montana, shows high antioxidant capacity and is reported to be an AMPK activator.

  • YN320001 NPS-2143 284035-33-2

    NPS-2143 is a novel potent and selective antagonist of Ca(2+) receptor with IC50 of 43 nM.

  • YN320185 NPS-2143 hydrochloride 324523-20-8

    NPS-2143 hydrochloride (SB-262470A hydrochloride), an orally active calcilytic agent, is a selective and potentcalcium ion-sensing receptor (CaSR)antagonist. NPS-2143 hydrochloride (SB-262470A hydrochloride) blocks increase...

  • YN321293 Cinacalcet hydrochloride 364782-34-3

    Cinacalcet HCl represents a new class of compounds for the treatment of hyperparathyroidism.

  • YN321284 Calcium-Sensing Receptor A... 478963-79-0

    Calcium-Sensing Receptor Antagonists I is an antagonist of calcium-sensing parathyroid hormone receptors.

  • YN321168 Evocalcet 870964-67-3

    Evocalcet has an activating effect oncalcium sensing receptor(CaSR) extracted from patent WO 2017061621 A1, compound A.

  • YN321988 Etelcalcetide hydrochloride 1334237-71-6

    Etelcalcetide hydrochloride (AMG 416 hydrochloride) is a synthetic peptide as an activator of thecalcium sensing receptor (CaSR). Etelcalcetide hydrochloride is effective in lowering parathyroid hormone (PTH) concentrations in ...

  • YN320253 Calhex 231 hydrochloride 2387505-78-2

    Calhex 231 hydrochloride is aCaSRinhibitor via negative allosteric modulation. Calhex 231 hydrochloride blocks Ca2+-induced accumulation of [3H]inositol phosphate with an IC50 of 0.39μM in HEK293 cells. Calhex 231 hydrochlori...

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