Calcitonin human is an endogenouscalcitonin receptoragonist.Calcitonin human lowers systemic blood calcium levels and inhibits bone resorption.
Salmon Calcitonin Acetate, which is more potent and longer lasting than human CT, has been used widely for the treatment of osteoporosis, paget's disease, hypercalcemic shock and chronic pain in terminal cancer patients.
PHM-27 (human) is a human prepro-vasoactive intestinal polypeptide (27 amino acid). PHM-27 (human) is a potent thehuman calcitonin receptoragonist with an EC50 of 11nM. PHM-27 (human) efficiently enhances glucose-induced insulin...
β-CGRP, human (Human β-CGRP) is one of calcitonin peptides, acts via the complex of calcitonin-receptor-like receptor (CRLR) and receptor-activity-modifying protein (RAMP), with IC50s of 1nM and 300nM for CRLR...
Adrenomedullin (AM) (22-52)...
Adrenomedullin (AM) (22-52), human, an NH2 terminal truncated adrenomedullin analogue, is anadrenomedullin receptorantagonist, and also antagonizes the calcitonin generelated peptide (CGRP) receptor in the hindlimb vascular bed o...
Kendomycin ((−)-TAN 2162) is a polyketideantibioticwith remarkable antibacterial and cancer cells cytotoxic activities. Kendomycin tends to be bacteriostatic rather than bactericidal and inhibits the growth of the methicillin-resi...
Olcegepant (BIBN-4096) is a potent and selective non-peptide antagonist of thecalcitonin gene-related peptide 1 (CGRP1) receptor with IC50 of 0.03nM and Kiof 14.4 pM for human CGRP.
Adrenomedullin (16-31), human
Adrenomedullin (16-31), human is amino acid residues 16-31 fragment of human adrenomedullin (hADM). Adrenomedullin has appreciable affinity for the CGRP1 receptor. Adrenomedullin (16-31), human possesses pressor activity in the sy...
Olcegepant hydrochloride (BIBN-4096 hydrochloride) is a potent and selective non-peptide antagonist of thecalcitonin gene-related peptide 1 (CGRP1) receptor with IC50 of 0.03nM and with a Ki of 14.4 pM for human CGRP.
Telcagepant (MK-0974) is an orally activecalcitonin gene-related peptide (CGRP) receptorantagonist with Kis of 0.77nM and 1.2nM for human and rhesus CGRP receptors, respectively.
MK-3207 (Hydrochloride) is a potent and orally bioavailableCGRP receptorantagonist with IC50 of 0.12nM and Kiof 0.024nM, and is highly selective versus human AM1, AM2, CTR, and AMY3.
MK-3207 is a potent and orally bioavailable CGRP receptor antagonist (IC50= 0.12nM; Ki value= 0.024nM); highly selective versus human AM1, AM2, CTR, and AMY3.
In common with other CGRP receptor antagonists, MK...
Rimegepant is a potent, selective, competitive human calcitonin gene-related peptide (CGRP) receptor antagonist with ki of 0.027 nM.
Ubrogepant (MK-1602) is a novel oral calcitonin gene-related peptide receptor (CGRP) antagonist in development for acute treatment of migraine.
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