Welcome to ULS!
Welcome to ULS!
> Products > Inhibitors & Agonists > GPCR/G Protein > CGRP Receptor
Products
CGRP Receptor

Chemical structure

Cat.No.

Product Name

CAS no.

Target

  • YN321991 Calcitonin (human) 21215-62-3

    Calcitonin human is an endogenouscalcitonin receptoragonist.Calcitonin human lowers systemic blood calcium levels and inhibits bone resorption.

  • YN321791 Calcitonin (salmon) 47931-85-1

    Salmon Calcitonin Acetate, which is more potent and longer lasting than human CT, has been used widely for the treatment of osteoporosis, paget's disease, hypercalcemic shock and chronic pain in terminal cancer patients.

  • YN321843 PHM-27 (human) 87403-73-4

    PHM-27 (human) is a human prepro-vasoactive intestinal polypeptide (27 amino acid). PHM-27 (human) is a potent thehuman calcitonin receptoragonist with an EC50 of 11nM. PHM-27 (human) efficiently enhances glucose-induced insulin...

  • YN321962 β-CGRP, human 101462-82-2

    β-CGRP, human (Human β-CGRP) is one of calcitonin peptides, acts via the complex of calcitonin-receptor-like receptor (CRLR) and receptor-activity-modifying protein (RAMP), with IC50s of 1nM and 300nM for CRLR...

  • YN321836 HCGRP-(8-37) 119911-68-1

    HCGRP-(8-37) is a human calcitonin gene-related peptide (hCGRP) fragment and also an antagonist ofCGRP receptor.

  • YN321809 Rat CGRP-(8-37) 129121-73-9

    Rat CGRP-(8-37) (VTHRLAGLLSRSGGVVKDNFVPTNVGSEAF) is a highly selectiveCGRP receptorantagonist.

  • YN321936 Adrenomedullin (AM) (22-52)... 159899-65-7

    Adrenomedullin (AM) (22-52), human, an NH2 terminal truncated adrenomedullin analogue, is anadrenomedullin receptorantagonist, and also antagonizes the calcitonin generelated peptide (CGRP) receptor in the hindlimb vascular bed o...

  • YN321975 Adrenomedullin (11-50), rat 163648-32-6

    Adrenomedullin (11-50), rat is the C-terminal fragment (11-50) of rat adrenomedullin. Rat adrenomedullin induces a selective arterial vasodilation via CGRP1 receptors.

  • YN320547 Kendomycin 183202-73-5

    Kendomycin ((−)-TAN 2162) is a polyketideantibioticwith remarkable antibacterial and cancer cells cytotoxic activities. Kendomycin tends to be bacteriostatic rather than bactericidal and inhibits the growth of the methicillin-resi...

  • YN320092 Olcegepant 204697-65-4

    Olcegepant (BIBN-4096) is a potent and selective non-peptide antagonist of thecalcitonin gene-related peptide 1 (CGRP1) receptor with IC50 of 0.03nM and Kiof 14.4 pM for human CGRP.

  • YN321977 Adrenomedullin (16-31), human 318480-38-5

    Adrenomedullin (16-31), human is amino acid residues 16-31 fragment of human adrenomedullin (hADM). Adrenomedullin has appreciable affinity for the CGRP1 receptor. Adrenomedullin (16-31), human possesses pressor activity in the sy...

  • YN320093 Olcegepant hydrochloride 586368-06-1

    Olcegepant hydrochloride (BIBN-4096 hydrochloride) is a potent and selective non-peptide antagonist of thecalcitonin gene-related peptide 1 (CGRP1) receptor with IC50 of 0.03nM and with a Ki of 14.4 pM for human CGRP.

  • YN321270 Telcagepant 781649-09-0

    Telcagepant (MK-0974) is an orally activecalcitonin gene-related peptide (CGRP) receptorantagonist with Kis of 0.77nM and 1.2nM for human and rhesus CGRP receptors, respectively.

  • YN320227 MK-3207 Hydrochloride 957116-20-0

    MK-3207 (Hydrochloride) is a potent and orally bioavailableCGRP receptorantagonist with IC50 of 0.12nM and Kiof 0.024nM, and is highly selective versus human AM1, AM2, CTR, and AMY3.

  • YN320225 MK-3207 957118-49-9

    MK-3207 is a potent and orally bioavailable CGRP receptor antagonist (IC50= 0.12nM; Ki value= 0.024nM); highly selective versus human AM1, AM2, CTR, and AMY3. In common with other CGRP receptor antagonists, MK...

  • YN320998 Rimegepant 1289023-67-1

    Rimegepant is a potent, selective, competitive human calcitonin gene-related peptide (CGRP) receptor antagonist with ki of 0.027 nM.

  • YN320579 Ubrogepant 1374248-77-7

    Ubrogepant (MK-1602) is a novel oral calcitonin gene-related peptide receptor (CGRP) antagonist in development for acute treatment of migraine.

    Contact

    TELL : +86-020-31703347

    Email: sales@ubiochem.com

    Add:Room 519, Block F, Guangzhou International Business Incubator, No.3 Lanyue Road, Science Town, Huangpu District, Guangzhou, China.

ULS products are chemical reagents for Research Use Only!Copyright © 2020-2021 ULS. All Rights Reserved.