Biochanin A, an O-methylated isoflavone from Trifolium pratense, inhibits protein tyrosine kinase (PTK) of epidermal growth factor receptor with IC50 values of 91.5 &muM.
URB597 is a potent, orally bioavailable FAAH inhibitor with IC50 of 4.6 nM, with no activity on other cannabinoid-related targets. Phase 1.
JNJ-1661010 is a potent and selective FAAH inhibitor with IC50 of 10 nM (rat) and 12 nM (human), exhibits >100-fold selectivity for FAAH-1 when compared to FAAH-2.
LY-2183240 is a potent, covalent inhibitor of the EC-degrading enzyme fatty acid amide hydrolase (FAAH). LY-2183240 disrupts the cellular uptake of the lipid endocannabinoid (EC) anandamide and promote analgesia in vivo. ...
N-Benzyloleamide is a maccamide isolated fromLepidium meyenii(Maca). N-Benzyloleamide irreversibly inhibits fatty acid amide hydrolase(FAAH). N-benzyloleamide influences the energy metabolism and reveals antioxidant and antif...
PF 750 is a selective and covalentfatty acid amide hydrolase (FAAH)inhibitor, with IC50 svaried from 16.2-595nM in different pre-incubation times. Covalently modifies the enzyme’s active site serine nucleophile.
PF-04457845 is a potent, favorable selective inhibitor of Fatty acid amide hydrolase (FAAH) with IC50 of 7.2 nM and 7.4 nM for hFAAH and rFAAH, respectively. PF-04457845 covalently modifies the active-site serine...
PF-3845 is a potent, selective and irreversible FAAH inhibitor with Ki of 230 nM, showing negligible activity against FAAH2.
BIA 10-2474 is a novel fatty acid amide hydrolase (FAAH) inhibitor, with a potent inhibitory effect upon FAAH and prolonged action in vivo.
SA57 is a potent, selectiveFAAHinhibitor with IC50s of 3.2nM and 1.9nM formouse and human FAAH. SA57 also inhibits the 2-arachidonoylglycerol hydrolasesMAGL(IC50s of 410nM and 1.4μM formouse and human MAG...
JNJ-42165279 (JNJ-5279) is an inhibitor of fatty acid amide hydrolase (FAAH) that inhibits recombinant human and rat FAAH with IC50 of 70 nM and 313 nM, respectively.
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