Ibrutinib Racemate (PCI-32765 Racemate) is the racemate of Ibrutinib. Ibrutinib is a selective, irreversibleBtkinhibitor with IC50 value of 0.5nM.
GDC-0834 Racemate is the racemate form of GDC-0834, which is a potent and selective BTK inhibitor with in vitro IC50s of 5.9 and 6.4nM in biochemical and cellular assays, respectively.
GDC-0834 is a potent and selectiveBTKinhibitor. GDC-0834 inhibits BTK with an in vitroIC50 of 5.9 and 6.4nM in biochemical and cellular assays, respectively, and in vivoIC50 of 1.1 and 5.6μM in mouse and rat, ...
Spebrutinib (CC-292, AVL-292) is a covalent, orally active, and highly selective BTK inhibitor with IC50 of <0.5 nM, displaying at least 1400-fold selectivity over the other kinases assayed. Phase 1.
CNX-500 is a probe consisting of a covalentBtkinhibitor (CC-292) chemically linked to biotin. CNX-500 retains inhibitory activity against Btk(IC50 of 0.5nM) and the ability to form a covalent bond withBtk. CNX-500 has low...
BMS-935177 is a potent, reversible Bruton's Tyrosine Kinase (BTK) inhibitor with an IC50 value of 2.8 nM and demonstrates good kinase selectivity. It is more potent against BTK than other kinase, including the other Tec fam...
CG-806 is an orally active, potent and non-covalent pan-FLT3/pan-BTKinhibitor with an IC50 of 0.08 µM forFLT3. CG-806 has an IC50 of 11nM againstFLT3wild type (WT)-transfected Ba/F3 cells.
(Rac)-IBT6A is a racemate of IBT6A. IBT6A is an impurity of Ibrutinib. IBT6A can be used in synthesis of IBT6A Ibrutinib dimer and IBT6A adduct. Ibrutinib is a selective, irreversible Btk inhibitor with an IC...
Acalabrutinib(ACP-196) is a selective second-generation Bruton's tyrosine kinase (BTK) inhibitor with an IC50 of 3 nM, which prevents the activation of the B-cell antigen receptor (BCR) signaling pathway. ACP-196 has impro...
Fenebrutinib (GDC-0853) is a potent, selective, orally available, and noncovalent bruton's tyrosine kinase (Btk) inhibitor with Kis of 0.91nM, 1.6, 1.3, 12.6, and 3.4nM for WT Btk, and the C481S, C481R, T474I, T474M...
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