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GHSR

Chemical structure

Cat.No.

Product Name

CAS no.

Target

  • YN320406 L-692429 145455-23-8

    L-692429 (MK-0751) is a benzolactam derivative and a nonpeptidylgrowth hormone secretagogue (GHS)agonist. L-692429 binds toG protein-coupled receptor with a Ki of 63nM.

  • YN321285 L-692585 145455-35-2

    L-692585 is a potent and nonpeptidylgrowth hormone secretagogue receptor (GHS-R1a)agonist, with a Ki of 0.8nM. L-692585 acts directly on somatotropes causing GH release.

  • YN321286 Ibutamoren Mesylate 159752-10-0

    Ibutamoren Mesylate (MK-677) is a potent, non-peptide Growth hormone secretagogue receptor (GHSR)agonist. Ibutamoren Mesylate is an orally active growth hormone (GH) secretagogue.

  • YN320949 Capromorelin Tartrate 193273-69-7

    Capromorelin Tartrate (CP 424391-18), a member of the growth hormone secretagogue (GHS) class of drugs, is a ghrelin receptor agonist and a novel therapy for stimulation of appetite in dogs with Ki of 7 nM for hGHS...

  • YN320901 Anamorelin 249921-19-5

    Anamorelin (ONO-7643, RC-1291, ST-1291) is an orally active, high-affinity, selective agonist of the ghrelin receptor with an EC50 value of 0.74 nM in the HEK293/GRLN FLIPR assay.

  • YN320902 Anamorelin hydrochloride 861998-00-7

    Anamorelin (RC-1291) hydrochloride is a potentghrelin receptoragonist withEC50value of 0.74nM in the FLIPR assay.

  • YN321901 Obestatin(rat) 869705-22-6

    Obestatin(rat), encoded by the Ghrelin gene, is a cpeptide, comprised of 23 amino acids. Obestatin(rat) suppresses food intake, inhibits jejunal contraction, and decreases body-weight gain. Obestatin is an endogenous lig and of G-pr...

  • YN321816 AZP-531 1088543-62-7

    AZP-531 is an analogue of unacylated ghrelin designed to improve glycaemic control and reduce weight.

  • YN320380 TM-N1324 1144477-35-9

    TM-N1324 is an agonist of G-Protein-Coupled Receptor 39 (GPR39) with EC50s of 9nM/5nM in the presence of Zn2+, and 280nM/180nM in the absence of Zn2+forhuman/murine GPR39.

  • YN320614 PF-5190457 1334782-79-4

    PF-5190457 (PF-05190457) is a potent and selectiveghrelin receptorinverse agonist with a pKi of 8.36.

  • YN320223 TC-G-1008 1621175-65-2

    TC-G-1008 (GPR39-C3) is a potent and orally available GPR39 agonist withEC50values of 0.4 and 0.8nM for rat and human receptors respectively.

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