Brilaroxazine
Cat. No. :YN320402
CAS No. :1239729-06-6
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5mg
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Product Name: | Brilaroxazine |
CAS NO.: | 1239729-06-6 |
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Molecular Weight: | 450.36 |
Molecular Formula: | C₂₂H₂₅Cl₂N₃O₃ |
SMILES: | O=C1NC2=CC(OCCCCN3CCN(C(C=CC=C4Cl)=C4Cl)CC3)=CC=C2OC1 |
Storage: | Please store the product under the recommended conditions in the Certificate of Analysis. |
Transportation: | Room temperature in continental US; may vary elsewhere. |
Description: | Brilaroxazine (RP5603) is a potent and orally active multimodaldopamine (DA)/serotonin (5-HT)modulator. Brilaroxazine is a partial agonist of dopamine (DA) D2, D3, and D4 receptors, 5-HT1A (Ki=1.5nM) and 5-HT2A (Ki=2.5nM), and has antagonist activity at 5-HT2B (Ki=0.19nM), and 5-HT7 (Ki=2.7nM) receptors. Brilaroxazine is an atypical antipsychotic agent, and has the potential to improve cognitive impairments in neuropsychiatric and neurological diseases in vivo. |
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