Grapiprant
Cat. No. :YN321095
CAS No. :415903-37-6
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order@ubiochem.com| Product Name: | Grapiprant |
| CAS NO.: | 415903-37-6 |
| Chemical Name: | |
| Synonyms: | |
| Molecular Weight: | 491.61 |
| Molecular Formula: | C₂₆H₂₉N₅O₃S |
| SMILES: | O=S(C1=CC=C(C)C=C1)(NC(NCCC2=CC=C(N3C(CC)=NC4=C3C=C(C)N=C4C)C=C2)=O)=O |
| Storage: | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Transportation: | Room temperature in continental US; may vary elsewhere. |
| Description: | Grapiprant (CJ-023423) is a selectiveEP4 receptorantagonist whose physiological lig and is prostagl and in E2(PGE2). Grapiprant displaces [3H]-PGE2(1nM) binding to dog recombinantEP4 receptor with IC50 value of 35nM and Kivalue of 24nM. Grapiprant has the potential for osteoarthritic pain and inflammation treatment . |
| IC50&Target: | |
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