Cligosiban
Cat. No. :YN320941
CAS No. :900510-03-4
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order@ubiochem.com| Product Name: | Cligosiban |
| CAS NO.: | 900510-03-4 |
| Chemical Name: | |
| Synonyms: | |
| Molecular Weight: | 419.84 |
| Molecular Formula: | C₁₉H₁₉ClFN₅O₃ |
| SMILES: | FC1=CC(Cl)=C(OC2CN(C3=NN=C(COC)N3C4=CC=C(OC)N=C4)C2)C=C1 |
| Storage: | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Transportation: | Room temperature in continental US; may vary elsewhere. |
| Description: | Cligosiban (PF-3274167), a high oral bioavailability and good brain-penetrant non-peptideoxytocin receptorantagonist, shows a high-affinity (Ki=9.5nM) and an excellent selectivity versus the vasopressin receptors with almost no affinity for the V1b and V1asubtypes. Cligosiban inhibits ejaculatory physiology in rodents. |
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