KG-501
Cat. No. :YN310061
CAS No. :18228-17-6
86-020-82000279
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order@ubiochem.com| Product Name: | KG-501 |
| CAS NO.: | 18228-17-6 |
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| Molecular Weight: | 377.72 |
| Molecular Formula: | C₁₇H₁₃ClNO₅P |
| SMILES: | O=C(C1=C(OP(O)(O)=O)C=C2C=CC=CC2=C1)NC3=CC=C(Cl)C=C3 |
| Storage: | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Transportation: | Room temperature in continental US; may vary elsewhere. |
| Description: | KG-501 is a cAMP response element-binding protein (CREB) inhibitor that disrupts CREB-dependent transcription (Ki = 10 μM) and CREB:CBP interaction (Ki = 50 μM). It also disrupts phospho (Ser-133) CREB binding to KIX with a Ki of ≈90 μM, using concentrations of CREB that were within the linear range of the binding assay. |
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