Apilimod mesylate
Cat. No. :YN330288
CAS No. :870087-36-8
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order@ubiochem.com| Product Name: | Apilimod mesylate |
| CAS NO.: | 870087-36-8 |
| Chemical Name: | |
| Synonyms: | STA-5326 mesylate |
| Molecular Weight: | 610.70 |
| Molecular Formula: | C₂₅H₃₄N₆O₈S₂ |
| SMILES: | CC1=CC=CC(/C=N/NC2=CC(N3CCOCC3)=NC(OCCC4=CC=CC=N4)=N2)=C1.CS(=O)(O)=O.CS(=O)(O)=O |
| Storage: | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Transportation: | Room temperature in continental US; may vary elsewhere. |
| Description: | Apilimod mesylate (STA-5326 mesylate) is a potent and orally-available inhibitor of the cytokines interleukin-12 (IL-12) and interleukin-23 (IL-23) with the potential to treat certain autoimmune and inflammatory diseases. Apilimod mesylate (STA-5326 mesylate) inhibits IL-12 with IC50 of 1 nM, 1 nM and 2 nM, in IFN-γ/SAC-stimulated human PBMCs, human monocytes and mouse PBMCs, respectively. Apilimod mesylate (STA-5326 mesylate) is also a cell permeable small molecule that specifically inhibits PIKfyve with IC50 of 14 nM. |
| IC50&Target: | |
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