PKC-IN-1
Cat. No. :YN310298
CAS No. :1046787-18-1
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Product Name: | PKC-IN-1 |
CAS NO.: | 1046787-18-1 |
Chemical Name: | |
Synonyms: | |
Molecular Weight: | 500.61 |
Molecular Formula: | C₂₅H₃₇FN₈O₂ |
SMILES: | O=C(N1[C@@H](C)CN(CC2CCOCC2)[C@H](C)C1)N(C3)C(C)(C)C4=C3C(NC5=NC(C)=NC=C5F)=NN4 |
Storage: | Please store the product under the recommended conditions in the Certificate of Analysis. |
Transportation: | Room temperature in continental US; may vary elsewhere. |
Description: | PKC-IN-1 is a potent, ATP-competitive and reversible inhibitor of conventionalPKCenzymes with Kis of 5.3 and 10.4nM for human PKCβ and PKCα, and IC50s of 2.3, 8.1, 7.6, 25.6, 57.5, 314, 808nM for PKCα, PKCβI, PKCβII, PKCθ, PKCγ, PKC mu and PKCε, respectively. |
IC50&Target: | |
In Vitro: | |
In Vivo: | |
Clinical Trial: | |
Solvent & Solubility: | |
References: |
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