GSK046
Cat. No. :YN310235
CAS No. :2474876-09-8
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order@ubiochem.com| Product Name: | GSK046 |
| CAS NO.: | 2474876-09-8 |
| Chemical Name: | |
| Synonyms: | iBET-BD2 |
| Molecular Weight: | 414.47 |
| Molecular Formula: | C₂₃H₂₇FN₂O₄ |
| SMILES: | O=C(N[C@H]1CC[C@H](O)CC1)C2=CC(O[C@H](C3=CC=CC=C3)C)=C(NC(C)=O)C(F)=C2 |
| Storage: | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Transportation: | Room temperature in continental US; may vary elsewhere. |
| Description: | GSK046 (iBET-BD2) is a selective and orally active inhibitor of BET (bromodomain and extraterminal domain) with IC50 of 264 nM, 98 nM, 49 nM and 214 nM for BRD2BD2, BRD3BD2, BRD4BD2 and BRDTBD2, respectively. GSK046 exhibits immunomodulatory activity. |
| IC50&Target: | |
| In Vitro: | |
| In Vivo: | |
| Clinical Trial: | |
| Solvent & Solubility: | |
| References: |
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