GS-6201
Cat. No. :YN1710001
CAS No. :752222-83-6
Pack size
price
inventory
10mg
$ 690.00
Product Name: | GS-6201 |
CAS NO.: | 752222-83-6 |
Chemical Name: | |
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Molecular Weight: | 446.43 |
Molecular Formula: | C₂₁H₂₁F₃N₆O₂ |
SMILES: | O=C(N1CCC)N(CC)C2=C(N=C(C3=CN(CC4=CC=CC(C(F)(F)F)=C4)N=C3)N2)C1=O |
Storage: | Please store the product under the recommended conditions in the Certificate of Analysis. |
Transportation: | Room temperature in continental US; may vary elsewhere. |
Description: | GS-6201 (CVT-6883) is a selectiveadenosine A2B receptorantagonist. GS-6201 displays high affinity and selectivity for the human adenosine A2B receptors (Ki=22nM). GS-6201 reduces caspase-1 activity in the heart, and attenuates cardiac remodeling after acute myocardial infarction (AMI) in the mouse. GS-62013 attenuates the airway reactivity induced by NECA, AMP, or allergen in sensitized mice. |
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References: |
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