SB-657510
Cat. No. :YN320306
CAS No. :474960-44-6
86-020-82000279
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order@ubiochem.com| Product Name: | SB-657510 |
| CAS NO.: | 474960-44-6 |
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| Molecular Weight: | 505.81 |
| Molecular Formula: | C₁₉H₂₂BrClN₂O₅S |
| SMILES: | ClC(C=C1)=C(O[C@H]2CN(C)CC2)C=C1NS(C3=CC(OC)=C(OC)C=C3Br)(=O)=O |
| Storage: | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Transportation: | Room temperature in continental US; may vary elsewhere. |
| Description: | SB-657510 is a selectiveurotensin II (UII) receptor (UT)antagonist. TheKivalues are 61, 17, 30, 65 and 56nM for human, monkey, cat, rat and mouse receptors, respectively. SB-657510 exerts anti-inflammatory effects by inhibiting UII-induced upregulation of inflammatory mediators such as adhesion molecules, cytokines, and tissue factor in human vascular endothelial cells. |
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