Ridaifen-B
Cat. No. :YN320214
CAS No. :886465-70-9
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price
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10mg
$ 680.00
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order@ubiochem.com| Product Name: | Ridaifen-B |
| CAS NO.: | 886465-70-9 |
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| Molecular Weight: | 510.71 |
| Molecular Formula: | C₃₄H₄₂N₂O₂ |
| SMILES: | CC/C(C1=CC=CC=C1)=C(C2=CC=C(OCCN3CCCC3)C=C2)C4=CC=C(OCCN5CCCC5)C=C4 |
| Storage: | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Transportation: | Room temperature in continental US; may vary elsewhere. |
| Description: | Ridaifen-B (RID-B) is a potent antagonist ofestrogen receptor α (ERα)with IC50 of 52.4nM, a tamoxifen (HY-13757A) derivative. Ridaifen-B is a high affinity, selective, inverse agonist atCB2receptor (Ki=43.7nM) over 17 foldsCB1receptor (Ki=732nM). Ridaifen-B modulates G-protein (IC50=300nM) and adenylyl cyclase activity with potency values predicted by CB2affinity (IC50=134nM). Ridaifen-B has anti-inflammatory, anti-cancer, and anti-osteoclastogenic effects. |
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