Gaboxadol hydrochloride
Cat. No. :YN360122
CAS No. :85118-33-8
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price
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5mg
$ 240.00
Product Name: | Gaboxadol hydrochloride |
CAS NO.: | 85118-33-8 |
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Molecular Weight: | 176.60 |
Molecular Formula: | C₆H₉ClN₂O₂ |
SMILES: | O=C1C2=C(CNCC2)ON1.Cl |
Storage: | Please store the product under the recommended conditions in the Certificate of Analysis. |
Transportation: | Room temperature in continental US; may vary elsewhere. |
Description: | Gaboxadol hydrochloride (Lu 02-030 hydrochloride; THIP hydrochloride) is a potent agonist of the GABAA receptor and an antagonist of GABAC receptors(IC50=25μM). Gaboxadol hydrochloride displays a partial agonist efficacy on subunit α1β2γ2 with an ED50 value of 143 µM, a full agonist efficacy at α5 subunit (ED50=28-129 µM) and a superagonist efficacy at α4β3δ (ED50=6 µM). Gaboxadol hydrochloride is a non-opioid analgesic and has hypnotic activities. |
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