GI-530159
Cat. No. :YN361092
CAS No. :69563-88-8
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price
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100mg
$ 50.00
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order@ubiochem.com| Product Name: | GI-530159 |
| CAS NO.: | 69563-88-8 |
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| Molecular Weight: | 518.45 |
| Molecular Formula: | C₂₇H₂₀F₆N₂O₂ |
| SMILES: | FC(C(C1=CC=C(OC2=CC=C(N)C=C2)C=C1)(C3=CC=C(OC4=CC=C(N)C=C4)C=C3)C(F)(F)F)(F)F |
| Storage: | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Transportation: | Room temperature in continental US; may vary elsewhere. |
| Description: | GI-530159 is a selective, mechanosensitive opener ofTREK1 (K2P2.1) and TREK2 (K2P10.1) channels, with an EC50 of 0.76μM for TREK1. GI-530159 displays selectivity for TREK1/2 over TRAAK, TASK3 and other potassium channels. GI-530159 reduces rat dorsal root ganglion neuron excitability. |
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