Azacyclonol
Cat. No. :YN481827
CAS No. :115-46-8
Pack size
price
inventory
500mg
$ 40.00
86-020-82000279
sales@ubiochem.com
order@ubiochem.com| Product Name: | Azacyclonol |
| CAS NO.: | 115-46-8 |
| Chemical Name: | |
| Synonyms: | |
| Molecular Weight: | 267.37 |
| Molecular Formula: | C₁₈H₂₁NO |
| SMILES: | OC(C1=CC=CC=C1)(C2CCNCC2)C3=CC=CC=C3 |
| Storage: | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Transportation: | Room temperature in continental US; may vary elsewhere. |
| Description: | Azacyclonol, also known as γ-pipradol, is a drug used to diminish hallucinations in psychotic individuals. Azacyclonol is a drug which is a so-called ataractive, or agent which diminishes hallucinations in psychotic individuals. The formation of Azacyclonol in human intestinal microsomes is linear with respect to time up to 60 min. The rates of formation of Azacyclonol increases linearly with microsomal protein concentration up to 2 mg/mL. The apparent Km and Vmax values of Azacyclonol are 0.82μM and 60 pmol/min/mg protein in microsomes from human liver . The formation of Azacyclonol and terfenadine alcohol from terfenadine is confirmed to be catalyzed predominantly by CYP3A(4) isozyme, and the ratio of the rate of terfenadine alcohol formation to that of Azacyclonol is 3:1 . The amount of Azacyclonol eliminated renally increases on average 2-fold after rifampin dosing . |
| IC50&Target: | |
| In Vitro: | |
| In Vivo: | |
| Clinical Trial: | |
| Solvent & Solubility: | |
| References: |
TELL : +86-020-82000279
Add:Room 519, Block F, Guangzhou International Business Incubator, No.3 Lanyue Road, Science Town, Huangpu District, Guangzhou, China.
