GSK2798745
Cat. No. :YN360692
CAS No. :1419609-94-1
86-020-82000279
sales@ubiochem.com
order@ubiochem.com| Product Name: | GSK2798745 |
| CAS NO.: | 1419609-94-1 |
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| Molecular Weight: | 460.53 |
| Molecular Formula: | C₂₅H₂₈N₆O₃ |
| SMILES: | N#CC1=CC=C2N=CN(C[C@](CCC3)(C)C[C@@]43CN(C5=NC=C(C(C)(O)C)N=C5)C(O4)=O)C2=C1 |
| Storage: | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Transportation: | Room temperature in continental US; may vary elsewhere. |
| Description: | GSK2798745 is a first-in-class, highly potent, selective, orally active transient receptor potential vanilloid 4(TRPV4) ion channelblocker with IC50s of 1.8 and 1.6nM for hTRPV4 and rTRPV4, respectively. GSK2798745 is used in research for the treatment of pulmonary edema associated with congestive heart failure. |
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