RPR-260243
Cat. No. :YN360594
CAS No. :668463-35-2
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order@ubiochem.com| Product Name: | RPR-260243 |
| CAS NO.: | 668463-35-2 |
| Chemical Name: | |
| Synonyms: | |
| Molecular Weight: | 510.50 |
| Molecular Formula: | C₂₈H₂₅F₃N₂O₄ |
| SMILES: | O=C([C@H]1CN(CC#CC2=CC(F)=CC(F)=C2F)CC[C@H]1CCC(C3=CC=NC4=CC=C(OC)C=C34)=O)O |
| Storage: | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Transportation: | Room temperature in continental US; may vary elsewhere. |
| Description: | RPR-260243, a potent activator ofhuman ether-a-go-go-related gene (hERG), slows deactivation and attenuates inactivation of hERG1 channels. RPR260243-modified HERG currents are inhibited by Dofetilide (IC50=58nM). RPR260243 displays no activator-like effects on other voltage-dependent ion channels, including the closely related ERG3 K+ channel. |
| IC50&Target: | |
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| Solvent & Solubility: | |
| References: |
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