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Glucocorticoid Receptor

Chemical structure

Cat.No.

Product Name

CAS no.

Target

  • YN321437 Desonide 638-94-8

    Desonide is a low potency topical corticosteroid.

  • YN321436 Meprednisone 1247-42-3

    Meprednisone is a glucocorticoid and a methylated derivative of prednisone.

  • YN321566 Betamethasone valerate 2152-44-5

    Betamethasone Valerate is a moderately potent glucocorticoid steroid with anti-inflammatory and immunosuppressive properties.

  • YN321653 Hydrocortisone hemisuccinate 2203-97-6

    Hydrocortisone hemisuccinate (A-hydrocort, Hydrocortisone 21-hemisuccinate), a physiological glucocorticoid with anti-inflammatory properties, is an inhibitor of proinflammatory cytokine with IC50 of 6.7 μM and 21.4 μM for <...

  • YN321683 Dexamethasone phosphate disod... 2392-39-4

    Dexamethasone phosphate disodium (DEX, Dexacort, Decadron, Dexair, Hexadrol, Maxidex) is a glucocorticoid receptor agonist with both anti-inflammatory and anti-oxidative effects.

  • YN321687 Methylprednisolone succinate 2921-57-5

    Methylprednisolone sodium succinate is a glucocorticoid used to treat a variety health issues including severe allergic reactions, asthma, autoimmune diseases, blood disorders, gastrointestinal diseases and endocrine disorders.

  • YN321615 Flunisolide 3385-03-3

    Flunisolide is a corticosteroid often used to treat allergic rhinitis.The principal mechanism of action of Flunisolide is to activate glucocorticoid receptors, meaning it has an anti-inflammatory action.

  • YN321620 Hydrocortisone phosphate 3863-59-0

    Hydrocortisone phosphate (Hydrocortisone 21-phosphate), a physiological glucocorticoid, and is an orally active steroidal anti-inflammatory drug (SAID). Hydrocortisone phosphate inhibits proinflammatory cytokine activity, with IC...

  • YN321664 Beclometasone 4419-39-0

    Beclometasone (Beclomethasone) is a prototypeglucocorticoid receptoragonist.

  • YN320543 Betamethasone acibutate 5534-05-4

    Betamethasone acibutate, derives from Betamethasone, is an acetate ester. Betamethasone acibutate is a glucocorticoid.

  • YN320758 Beclometasone dipropionate 5534-09-8

    Beclomethasone dipropionate is a potent glucocorticoid steroid used for the treatment of rhinitis and sinusitis.

  • YN320768 Beclomethasone 17-propionate 5534-18-9

    Beclomethasone 17-propionate (Beclomethasone-17-monopropionate), an active metabolite of Beclomethasone dipropionate (HY-13571), is aglucocorticoid receptor (GR)agonist. Beclomethasone 17-propionate exhibits greater affinity for GR...

  • YN320757 Betamethasone dipropionate 5593-20-4

    Betamethasone Dipropionate is a glucocorticoid steroid with anti-inflammatory and immunosuppressive abilities.

  • YN322024 Prednisolone Tebutate 7681-14-3

    Prednisolone tebutate is a synthetic glucocorticoid used as an antiinflammatory and immunosuppressant.

  • YN320395 Vamorolone 13209-41-1

    Vamorolone (VBP15) is a first-in-class, orally activedissociative steroidal anti-inflammatorydrug and membrane-stabilizer. Vamorolone improves muscular dystrophy without side effects. Vamorolone shows potentNF-κBinhibition and ...

  • YN320764 Deflazacort 14484-47-0

    Deflazacort is a glucocorticoid used as an anti-inflammatory and immunosuppressant.

  • YN320664 Dexamethasone palmitate 14899-36-6

    Dexamethasone palmitate (DXP), a lipophilic prodrug of Dexamethasone (DXM), is a glucocorticoid receptor agonist with a 47-fold lower affinity for the glucocorticoid receptor than DXM. Dexamethasone palmitate (DXP) exh...

  • YN321670 Clobetasone butyrate 25122-57-0

    Clobetasone butyrate is a new corticosteroid that is often employed topically as a treatment for a variety of conditions such as eczema, psoriasis, various forms of dermatitis, and also for certain ophthalmologic conditions.

  • YN322013 Triamcinolone Benetonide 31002-79-6

    Triamcinolone benetonide is a synthetic glucocorticoid corticosteroid with anti-inflammatory activity.

  • YN321735 (20S)-Protopanaxatriol 34080-08-5

    (20S)-Protopanaxatriol(g-PPT), a neuroprotective metabolite of ginsenoside, protopanaxatriol (g-PPT), is a functional ligand for both GR and ERbeta and could modulate endothelial cell functions through the glucocorticoid recepto...

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