ELN-441958
Cat. No. :YN320943
CAS No. :913064-47-8
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Product Name: | ELN-441958 |
CAS NO.: | 913064-47-8 |
Chemical Name: | |
Synonyms: | |
Molecular Weight: | 501.02 |
Molecular Formula: | C₂₉H₂₉ClN₄O₂ |
SMILES: | ClC1=C2C(CN(C3=CC=CC(C(N4CCC5(CCN(C6=CC=NC=C6)CC5)CC4)=O)=C3)C2=O)=CC=C1 |
Storage: | Please store the product under the recommended conditions in the Certificate of Analysis. |
Transportation: | Room temperature in continental US; may vary elsewhere. |
Description: | ELN-441958 is a potent, neutral antagonist of B1 receptor, inhibits the binding of the B1 agonist lig and [3H]DAKD to IMR-90 cells with Ki of 0.26nM. ELN-441958 is highly selective for B1 over B2 receptors, and >500/ 2000-fold selective for the B1 over μ/δ-opioid receptor. |
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References: |
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