Nebentan
Cat. No. :YN320311
CAS No. :403604-85-3
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order@ubiochem.com| Product Name: | Nebentan |
| CAS NO.: | 403604-85-3 |
| Chemical Name: | |
| Synonyms: | |
| Molecular Weight: | 491.52 |
| Molecular Formula: | C₂₄H₂₁N₅O₅S |
| SMILES: | O=S(/C=C/C1=CC=CC=C1)(NC2=NC(C3=NC=CC=N3)=NC(OC)=C2OC4=CC=CC=C4OC)=O |
| Storage: | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Transportation: | Room temperature in continental US; may vary elsewhere. |
| Description: | Nebentan (YM598 free base) is a potent, selective and orally active non-peptideendothelin ETAreceptorantagonist through the modification of Bosentan (HY-A0013). Nebentan inhibits [125I] endothelin-1 binding to cloned human endothelin ETA and ETB receptor, with Kiof 0.697nM and 569nM, respectively. YM598 can ameliorate the progression of cor pulmonale and myocardial infarction in vivo. |
| IC50&Target: | |
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