YN250877 Cilastatin sodium 81129-83-1

Cilastatin sodium (MK0791 sodium) is a reversible, competitiverenal dehydropeptidase Iinhibitor with an IC50 of 0.1μM. Cilastatin sodium inhibits thebacterial metallob-lactamase enzyme CphAwith an IC50 of 178μM. Cilastatin s...

YN250378 Acetyllovastatin 81189-92-6

Acetyllovastatin, a acetate of Lovastatin, presentes a moderate inhibitory effect againstthe enzyme acetylcholinesterasewith an IC50 of 79 μg/mL. Lovastatin has been found to display antifungal activity, and suppresses proliferatio...

YN250294 Caracemide 81424-67-1

Caracemide (NSC-253272) inhibits the enzymeribonucleotide reductaseof Escherichia coli. Caracemide is a novel anticancer agent derived from a hydroxamic acid and has demonstrated to produce severe central nervous system (CNS) tox...

YN330001 Peretinoin 81485-25-8

Peretinoin is an oral acyclic retinoid retinoid with a vitamin A-like structure that targets retinoid nuclear receptors such asretinoid X receptor(RXR) and retinoic acid receptor (RAR).

YN250339 Quinocetone 81810-66-4

Quinocetone is a potent synthetic antimicrobial agent that is used for improving the feed efficiency and controlling dysentery in food-producing animals.

YN372280 Vesnarinone 81840-15-5

Vesnarinone is a quinolinone derivative, and its pharmacodynamic effects include inhibition of phosphodiesterase III (PDE3) activity, increases in calcium flux and decreases in potassium flux.

YN373234 Ganoderic acid B 81907-61-1

Ganoderic acid B is a triterpene isolated from a mushroomGanoderma lucidum. Ganoderic acid B inhibits the activation of Epstein-Barr virus (EBV) antigens as telomerase inhibitor. Ganoderic acid B is a moderately active inhibitor...

YN251483 (Z)-Ligustilide 81944-09-4

(Z)-Ligustilide is extracted fromLigusticum chuanxiong Hort, has antimicrobial and antifungal activity, exhibits an average antifungal score of 5.6. (Z)-Ligustilide inhibits the expression of FATP5 and DGAT, inhibits fatty...

YN250876 Cilastatin 82009-34-5

Cilastatin is a renal dehydropeptidase-I and leukotriene D4 dipeptidase inhibitor.

YN321119 Loteprednol Etabonate 82034-46-6

Loteprednol etabonate is a potent glucocorticoid receptor agonist, used in treatment of inflammation of the eye due to allergies.

YN251722 Ludaconitine 82144-72-7

Ludaconitine, isolated fromAconitum spicatum(Bruhl) Stapf, exhibits antileishmanial activity with an IC50 of 36.10 μg/mL.

YN251135 Lumefantrine 82186-77-4

Lumefantrine is an antimalarial agent used to treat acute uncomplicated malaria.

YN250323 Ansatrienin B 82189-04-6

Ansatrienin B (Mycotrienin II) is an ansamycinantibioticisolated fromStreptomyces. Ansatrienin B is active against fungi and yeasts, but inactive against bacteria.Ansatrienin B displays antitumor antibiotic activity and can be...

YN251325 Sulconazole nitrate 82382-23-8

Sulconazole nitrate ((±)-Sulconazole nitrate), an imidazole derivative, is a broad-spectrum fungicide and is inhibitory to certain gram-positive anaerobes. Sulconazole nitrate can be used for the research of dermatomycoses, pityriasis...

YN250528 Ganciclovir 82410-32-0

Ganciclovir is an antiviral drug for feline herpesvirus type-1 with IC50 of 5.2 μM in a cell-free assay.

YN250916 Ofloxacin 82419-36-1

Ofloxacin is a synthetic broad-spectrum antimicrobial agent.

YN251642 Gomisin M2 82425-45-4

Gomisin M2 ((+)-Gomisin M2) is a lignan isolated from the fruits ofSchis and ra rubriflorawith anti-HIVactivity (EC50of 2.4μM). Gomisin M2 exhibits anti-cancer and anti-allergic activities and has the potential for Alzhei...

YN251731 Pseudolaric Acid B 82508-31-4

Pseudolaric acid B, a natural diterpenoid compound, is isolated from Pseudolarix kaempferi.

YN251517 Pseudolaric Acid A 82508-32-5

Pseudolaric Acid A is a diterpene acid isolated fromPseudolarix kaempferi, has antifungal, cytotoxic and antifertile activities .

YN250134 Cefteram pivoxil 82547-81-7

Cefteram pivoxil (Ro 19-5248), an orally active cephalosporin antibiotic, is used for bacterial infections.