YN250197 Tafenoquine Succinate 106635-81-8

Tafenoquine Succinate (WR 238605 Succinate) is an 8-aminoquinoline. Tafenoquine is an anti-malarial prophylactic agent.

YN251364 Adefovir 106941-25-7

Adefovir (GS-0393) is an adenosine monophosphate analog antiviral agent that after intracellular conversion to Adefovir diphosphate inhibitsHBVDNA polymerase. Adefovir has an IC50 of 0.7μM againstHBVin the HepG2.2.15 cel...

YN372863 Tebuconazole 107534-96-3

Tebuconazole is an agricultural azole fungicide which can also inhibitCYP51with IC50s of 0.9 and 1.3μM forC and ida albicansCYP51 (CaCYP51) and truncatedHomo sapiensCYP51 (Δ60HsCYP51), respectively.

YN250784 4-Phenoxybenzylamine 107622-80-0

4-Phenoxybenzylamine inhibits the function of theNS3protein by stabilizing an inactive conformation with an IC50 of about 500μM against FL NS3/4a.

YN373309 Ganodermanondiol 107900-76-5

Ganodermanondiol is a melanogenesis inhibitor isolated from theGanoderma lucidum.Ganodermanondiol exhibits potent cytoprotective effects on tert-butyl hydroperoxide-induced hepatotoxicity. Ganodermanondiol shows significant anti-HIV-...

YN250529 Ganciclovir sodium 107910-75-8

Ganciclovir sodium is an antiviral medication used to treat cytomegalovirus (CMV) infections

YN251162 Tilmicosin 108050-54-0

Tilmicosin is a macrolide antibiotic.

YN251714 KT5720 108068-98-0

KT5720 is a cell-permeable, potent, specific, reversible, ATP-competitive inhibitor ofprotein kinase A (PKA), with a Ki of 60nM.

YN250810 Calicheamicin 108212-75-5

Calicheamicin, anantitumor antibiotic, is a cytotoxic agent that causes double-str and DNA breaks. Calicheamicin is a DNA synthesisinhibitor.

YN251807 Magainin 2 108433-95-0

Magainin 2 (Magainin II) is anantimicrobial peptide (AMP)isolated from the skin of the African clawed frogXenopus laevis. Magainin 2 displays antibiotic activity against numerous gram-negative and gram-positive bacteria. Magai...

YN251806 Magainin 1 108433-99-4

Magainin 1 (Magainin I) is an antimicrobial and amphipathic peptide isolated from the skin ofXenopus laevis. Magainin 1 exhibits antibiotic activity against numerous Gram-negative and Gram-positivebacteria .

YN250564 Tacrolimus monohydrate 109581-93-3

Tacrolimus monohydrate (FK506 monohydrate), a macrocyclic lactone, binds toFK506 binding protein (FKBP)to form a complex and inhibitscalcineurin phosphatase, which inhibits T-lymphocyte signal transduction and IL-2 transcrip...

YN320048 Plerixafor 110078-46-1

Plerixafor (AMD3100) is a chemokine receptor antagonist for CXCR4 and CXCL12-mediated chemotaxis with IC50 of 44 nM and 5.7 nM in cell-free assays, respectively.

YN371561 4-Desmethoxy Omeprazole 110374-16-8

4-Desmethoxy Omeprazole is the active metabolite of Omeprazole. Omeprazole, a proton pump inhibitor (PPI), is available for treatment of acid-related gastrointestinal disorders. Omeprazole shows competitive inhibition of CYP2C19...

YN251888 Saperconazole 110588-57-3

Saperconazole (R66905) is a broad-spectrumantifungaltriazole and has potent activity againstAspergilluswith anMIC90of 0.19 mg/L.

YN251583 Psammaplin A 110659-91-1

Psammaplin A, a marine metabolite, is a potent inhibitor ofHDAC and DNA methyltransferases. Psammaplin A ia a highly potent and selectiveDAC1inhibitor with an IC50 of 0.9nM. Psammaplin A possess the antimicrobial effect...

YN250994 Sparfloxacin 110871-86-8

Sparfloxacin is a fluoroquinolone antibiotic, shows broad and potent antibacterial activity.

YN250399 Okilactomycin 111367-04-5

Okilactomycin is a lactone groupantibioticisolated from the culture filtrate of a strain of actinomycetes (Streptomyces species).

YN340202 Ochromycinone 111540-00-2

Ochromycinone (STA-21) is a selective STAT3 inhibitor.

YN251375 Cefetamet pivoxil hydrochlori... 111696-23-2

Cefetamet pivoxil hydrochloride is the hydrochloride salt form of cefetamet pivoxil, which is an oral third-generation cephalosporin antibiotic.