MK-2 Inhibitor III
Cat. No. :YN350083
CAS No. :1186648-22-5
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order@ubiochem.com| Product Name: | MK-2 Inhibitor III |
| CAS NO.: | 1186648-22-5 |
| Chemical Name: | |
| Synonyms: | |
| Molecular Weight: | 358.39 |
| Molecular Formula: | C₂₁H₁₈N₄O₂ |
| SMILES: | O=C1C2=C(NC(C3=CC(C4=CC5=CC=CC=C5N=C4)=NC=C3)=C2)CCN1.O |
| Storage: | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Transportation: | Room temperature in continental US; may vary elsewhere. |
| Description: | MK-2 Inhibitor III (compound 16) is an orally active, selective, and ATP-competitiveMAPKAP-K2 (MK-2)inhibitor with an IC50 of 0.85nM, and is exceptional selectivity against MK-3 (IC50=0.21μM), MK-5 (IC50=0.081μM), ERK2 (IC50=3.44μM), MNK1(IC50=5.7μM) as well as CDK2, JNK2, IKK2, MSK1, and MSK2. |
| IC50&Target: | |
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