Chemical structure
Cat.No.
Product Name
CAS no.
Target
YN322017 Cicloprolol hydrochloride 63686-79-3
Cicloprolol is a partialβ 1-adrenoceptoragonist .
YN321418 Tizanidine hydrochloride 64461-82-1
Tizanidine HCl is an α2-adrenergic receptor agonist and inhibits neurotransmitter release from CNS noradrenergic neurons.
YN322081 Bometolol Hydrochloride 65023-16-7
Bometolol Hydrochloride is abeta-adrenergicblocking agent, used for the research of cardiovascular disease.
Teoprolol is aβ-adrenergic receptorblocker.
YN320666 Bisoprolol 66722-44-9
Bisoprolol is a cardioselective β1-adrenergic blocking agent used for secondary prevention of myocardial infarction (MI), heart failure, angina pectoris and mild to moderate hypertension.
YN320021 Tiodazosin 66969-81-1
Tiodazosin is a potent competitive postsynapticalpha adrenergic receptorantagonist.
YN321465 Terazosin hydrochloride dihyd... 70024-40-7
Terazosin HCl is a selective α1-adrenoceptor antagonist, used for treatment of symptoms of an enlarged prostate (BPH).
YN321552 Brimonidine tartrate 70359-46-5
Brimonidine Tartrate is a highly selective α-adrenergic receptor agonist with EC50 of 0.45 nM for the α2A adrenoreceptor, and used to treat open-angle glaucoma or ocular hypertension.
YN320250 Bucindolol 71119-11-4
Bucindolol is aβ1-adrenergic receptorblocker, with intrinsic sympathomimetic activity, used in the research of heart failure.
D2343 is aβ2-adrenoceptoragonist and also is anα1- adrenoceptorinhibitor.
YN320811 ICI 118,551 hydrochloride 72795-01-8
ICI 118,551 (hydrochloride) is a highly selectiveβ2 adrenergic receptorantagonist, with Kis of 0.7, 49.5 and 611nM for β2, β1 and β3 receptors, respectively.
YN321355 Dapiprazole hydrochloride 72822-13-0
Dapiprazole Hydrochloride is the hydrochloride salt form of dapiprazole, an alpha-adrenergic blocker used to reverse mydriasis after eye examination.
YN321368 Carvedilol 72956-09-3
Carvedilol is a non-selective beta blocker/alpha-1 blocker, used to treat congestive heart failure (CHF) and high blood pressure.
Doxazosin is a quinazoline-derivative that selectively antagonizes postsynaptic α1-adrenergic receptors.
Ro 363 is a potent and highly selectiveβ1-adrenoceptoragonist. RO 363 is an effective inotropic stimulant, and is a cardiovascular modulator that reduces diastolic blood pressure and pronounces increases in myocardial contractilit...
Ancarolol is abeta-adrenergicblocking agent.
YN321402 Detomidine 76631-46-4
Detomidine, an imidazole derivative, is a potentα2-adrenergicagonist. Detomidine produces dose-dependent sedative and analgesic effects.
Ecastolol is abeta adrenergic receptorantagonist, with antianginal activities.
YN321387 Doxazosin mesylate 77883-43-3
Doxazosin, a quinazoline-derivative, selectively antagonizes postsynaptic α1-adrenergic receptors, used in the treatment of high blood pressure and urinary retention associated with benign prostatic hyperplasia.
YN320777 Bromchlorbuterol hydrochlorid... 78982-84-0
Bromchlorbuterol hydrochloride is an active β-adrenergic agonist (β-agonist) and can be used for the research of pulmonary disease and asthma.
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