YN321654 Efaroxan hydrochloride 89197-00-2

Efaroxan hydrochloride is a potent and selectiveα2-adrenoceptorantagonist, with antidiabetic activity. Efaroxan hydrochloride is a selectiveI1-Imidazoline receptorantagonist and can be used for the research of cardiovascular diseas...

YN320848 Salmeterol 89365-50-4

Salmeterol is a long-acting beta2-adrenergic receptor agonist with Ki value of 1.5 nM for WT β2AR and shows very high selectivity for the WT β2AR(β1Ki/β2Ki ratio of approximately 1500).

YN321403 Detomidine hydrochloride 90038-01-0

Detomidine hydrochloride, an imidazole derivative, is a potentα2-adrenergicagonist. Detomidine hydrochloride produces dose-dependent sedative and analgesic effects.

YN320065 Hydroxybupropion 92264-81-8

Hydroxybupropion is the major active metabolite of Bupropion. Hydroxybupropion is metabolized by CYP2B6.Bupropion is an atypical antidepressant and smoking-cessation agent. Hydroxybupropion inhibitsnorepinephrine uptakewith an I...

YN320200 Naminterol 93047-40-6

Naminterol is a phenethanolamine derivative, is aβ2adrenoceptoragonist with bronchodilatory properties. Naminterol is used for treatment of asthma.

YN321583 Nadolol D9 94513-92-5

Nadolol D9 (SQ-11725 D9) is the deuterium labeled Nadolol. Nadolol is a non-selective and orally activeβ-adrenergic receptorsblocker.

YN321139 Salmeterol xinafoate 94749-08-3

Salmeterol xinafoate is a long-acting beta-2 adrenergic receptor (β2AR) agonist, with Kiof 1.5nM for WT β2AR, and used for asthma treatment.

YN321371 (R)-Carvedilol 95093-99-5

(R)-Carvedilol ((R)-BM 14190), the R-enantiomer of Carvedilol, is a non-selectiveβ/α-1blocker. (R)-Carvedilol exerts protection against the vascular or cardiac toxicity of Doxorubicin (DOX).

YN321370 (S)-Carvedilol 95094-00-1

(S)-Carvedilol, the S-enantiomer of Carvedilol, is a non-selectiveβ/α-1blocker. (S)-Carvedilol exerts protection against the vascular or cardiac toxicity of Doxorubicin (DOX).

YN321153 Metoprolol Succinate 98418-47-4

Metoprolol Succinate (Toprol XL) is a selective β1 receptor blocker used in treatment of several diseases of the cardiovascular system, especially hypertension.

YN320585 Atipamezole 104054-27-5

Atipamezole is a synthetic α2 adrenergic receptor antagonist. It has also been researched in humans as a potential anti-Parkinsonian drug.

YN320584 Atipamezole hydrochloride 104075-48-1

Atipamezole is a synthetic α2 adrenergic receptor antagonist. It has also been researched in humans as a potential anti-Parkinsonian drug. Atipamezole hydrochloride is hydrochloride form of atipamezole.

YN321385 (±)-Bisoprolol hemifumarate 104344-23-2

Bisoprolol fumarate is a selective type β1 adrenergic receptor blocker.

YN320134 CGP 20712 A 105737-62-0

CGP 20712 A (CGP 20712 mesylate) is a highly selectiveβ1-adrenoceptorantagonist with an IC50 of 0.7nM. CGP 20712 A exhibits ~10,000-fold selectivity over β2-adrenoceptors.

YN321553 Tamsulosin 106133-20-4

Tamsulosin is a selective α1 receptor antagonist that has preferential selectivity for the α1A receptor in the prostate versus the α1B receptor in the blood vessels.

YN322056 Falintolol, (Z)- 106401-52-9

Falintolol, (Z)-, a newβ-adrenergicantagonist, is characterized by the presence of an oxime function.

YN321554 Tamsulosin hydrochloride 106463-17-6

Tamsulosin (Flomax) hydrochloride is an antagonist of alpha1A adrenoceptors in the prostate.

YN320795 Norepinephrine bitartrate mon... 108341-18-0

Noradrenaline bitartrate monohydrate is a direct alpha-adrenergic receptors stimulator.

YN321467 (S)-Terazosin 109351-33-9

(S)-Terazosin is an active S-enantiomer of Terazosin. (S)-Terazosin is a potent and high-affinityα-adrenoceptorantagonist with Ki values of 3.91nM, 0.79nM and 1.16nM forα1a,α1b and α1d-adrenoceptor, respectively. (S)-Ter...

YN321466 (R)-Terazosin 109351-34-0

(R)-Terazosin is an active R-enantiomer of Terazosin. (R)-Terazosin is a potentα1-adrenoceptorantagonist with Ki values of 6.51nM, 1.01nM and 1.97nM forα1a,α1b and α1d-adrenoceptor, respectively.