YN250743 Bethoxazin 163269-30-5

Bethoxazin(Bethoguard) is a new broad spectrum industrial microbicide with applications in material and coating preservation. Bethoxazin potently inhibited the catalytic activity of yeast DNA topoisomerase II and the growth of y...

YN251123 Pazufloxacin mesylate 163680-77-1

Pazufloxacin Mesylate, also known as Pazucross and T-3762, is a quinolone antibacterial agent used for the intravenous therapy of several infections.

YN250649 Efinaconazole 164650-44-6

Efinaconazole is an inhibitor of 14 alpha-demethylase which is involved in the biosynthesis of ergosterol, a constituent of fungal cell membranes.

YN360840 Dinotefuran 165252-70-0

Dinotefuran is an insecticide of the neonicotinoid class, its mechanism of action involves disruption of the insect's nervous system by inhibiting nicotinic acetylcholine receptors.

YN250097 Linezolid 165800-03-3

Linezolid is a synthetic antibiotic used for the treatment of serious infections.

YN250096 Eperezolid 165800-04-4

Eperezolid(PNU-100592) is a oxazolidinone antibacterial agent, Eperezolid demonstrated good in vitro inhibitory activity, regardless of methicillin susceptibility for staphylococci(MIC90= 1-4 mg/ml).

YN372531 PNU-103017 166335-18-8

PNU-103017 is anHIV proteaseinhibitor.

YN250545 Tenofovir diphosphate 166403-66-3

Tenofovir diphosphate (TFV-DP) is a competitiveDNA polymerasesinhibitor (with respect to dATP) and a substrate of HIV type 1 (HIV-1)reverse transcriptase(RT).

YN250491 Anidulafungin 166663-25-8

Anidulafungin (LY303366), an echinocandin derivative, inhibits glucan synthase activity, used as an antifungal drug.

YN250791 Ornidazole (Levo-) 166734-83-4

Ornidazole Levo- is the levo-isomer of Ornidazole. Ornidazole is a 5-nitroimidazole derivative with antiprotozoal and antibacterial properties against anaerobic bacteria. Ornidazole Levo- is the less active isomer.

YN251629 Triptonine B 168009-85-6

Triptonine B, a sesquiterpene pyridine alkaloid that isolated fromTripterygium hypoglaucum and Tripterygium wilfordii, inhibitsHIVreplication in H9 lymphocytes with an EC50 value of <0.10 μg/mL.

YN320821 Rimonabant 168273-06-1

Rimonabant is a selective antagonist of CB1 with IC50 of 13.6 nM and EC50 of 17.3 nM in hCB1 transfected HEK 293 membrane.

YN250095 Sutezolid 168828-58-8

Sutezolid (PNU-100480), an orally active oxazolidinone antimicrobial agent, acts by inhibitingbacterial protein synthesis. Sutezolid has potent activity againstmycobacteria, and is used for the research of drug-resistant tuberculosis...

YN250550 Demethyl linezolid 168828-65-7

Demethyl linezolid is a impurity of linezolid. Demethyl linezolid is a useful antimicrobial agent extracted from patent WO1995007271A1, example 9, effective against a number of human and veterinary pathogens.

YN250009 Fluazinam impurity 1 169327-87-1

Fluazinam impurity 1 is an impurity of Fluazinam with antifungal activity. Fluazinam impurity 1 is active againstSphaerotheca fuliginea,Pyricularia oryzae and Rhizoctonia solani.

YN250021 AQ-13 dihydrochloride 169815-40-1

AQ-13 dihydrochloride is an aminoquinoline antimalarial drug that is effective against drug-resistant strains ofPlasmodium falciparum.

YN250070 Antibacterial compound 2 170104-58-2

Antibacterial compound 2 is a usefulantibacterialagent extracted from patent US5652238, compound example 9.

YN371186 LHVS 170111-28-1

LHVS is a potent, non-selectivecysteine proteaseinhibitor. LHVS effectively blocksT. gondiimicroneme protein secretion (IC50=10μM), gliding motility, and cell invasion.

YN340136 AG-1478 hydrochloride 170449-18-0

AG-1478 hydrochloride (Tyrphostin AG-1478 hydrochloride) is a selectiveEGFRtyrosine kinase inhibitor with IC50 of 3nM. AG-1478 hydrochloride has antiviral effects againstHCV and encephalomyocarditis virus (EMCV).

YN250702 Posaconazole 171228-49-2

Posaconazole is an inhibitor primarily of CYP3A4, but it does not inhibit the activity of other CYP enzymes Also an inhibitor of sterol C14ɑ demethylase inhibitor with IC50 of 0.25 μM. Posaconazole has a median terminal elim...