Sapitinib
Cat. No. :YN340121
CAS No. :848942-61-0
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order@ubiochem.com| Product Name: | Sapitinib |
| CAS NO.: | 848942-61-0 |
| Chemical Name: | |
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| Molecular Weight: | 473.93 |
| Molecular Formula: | C₂₃H₂₅ClFN₅O₃ |
| SMILES: | O=C(CN1CCC(OC2=CC3=C(NC4=CC=CC(Cl)=C4F)N=CN=C3C=C2OC)CC1)NC |
| Storage: | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Transportation: | Room temperature in continental US; may vary elsewhere. |
| Description: | Sapitinib (AZD8931) is a reversible, ATP competitive inhibitor of EGFR, ErbB2 and ErbB3 with IC50 of 4 nM, 3 nM and 4 nM in cell-free assays, more potent than Gefitinib or Lapatinib against NSCLC cell, 100-fold more selective for the ErbB family than MNK1 and Flt. Phase 2. |
| IC50&Target: | |
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