Chemical structure
Cat.No.
Product Name
CAS no.
Target
YN250355 Epetraborole hydrochloride 1234563-16-6
Epetraborole hydrochloride is a novel leucyl-tRNA synthetase (LeuRS) inhibitor, which inhibits protein synthesis by binding "to the terminal adenosine ribose (A76) of leucyl-tRNA synthetase". It is intended for the treatment of ...
TBA-354 is a potent anti-tuberculosis compound; maintains activity against Mycobacterium tuberculosis H37Rv isogenic monoresistant strains.
YN251075 Amikacin hydrate 1257517-67-1
Amikacin is an aminoglycoside antibiotic used to treat different types of bacterial infections.
YN250779 MUT056399 1269055-85-7
MUT056399 (Fab-001) is a highly potent inhibitor of the FabI enzymeof both S. aureus and E. coli with 50% inhibitory concentrationIC50s of 12nM and 58nM, respectively.
YN251178 Sulfamonomethoxine D4 1286538-12-2
Sulfamonomethoxine D4 is a deuterium labeled Sulfamonomethoxine. Sulfamonomethoxine is a long acting sulfonamide antibacterial agent, used in blood kinetic studies, and blocks the synthesis of folic acid by inhibiting synthetase of dih...
Q203 (IAP6) is a midazopyridine amide compound. Q203 is active against Mycobacterium tuberculosisH37Rv with an MIC50 of 2.7nM in culture broth medium.
AU1235, an adamantyl urea, is a potent inhibitor of Mycobacterium tuberculosis protein MmpL3.
YN250685 Lefamulin acetate 1350636-82-6
Lefamulin acetate (Xenleta, BC-3781 acetate) is a pleuromutilin antibiotic for community-acquired bacterial pneumonia (CABP) treatment. Lefamulin acetate inhibits protein synthesis by binding to the peptidyl transferase c...
YN251614 Isoforsythiaside 1357910-26-9
Isoforsythiaside, isolated fromForsythia suspensa, is an antioxidant and antibacterial phenylethanoid glycoside with MICs of 40.83, 40.83, and 81.66 μg/mL forEscherichia coli(E. coli),Pseudomonas aeruginosa(PAO), and Stap...
YN250198 (3R,4R)-A2-32-01 1359752-95-6
(3R,4R)-A2-32-01 (compound 2), an anti-virulence drug, is a specificcaseinolytic protein proteases (ClpP)inhibitor with an EC50 of 4.5μM, and shows a tolerable cytotoxicity.
M4284 is a selective and orally active biphenyl mannosideFimHantagonist. M4284 has activities against different UPEC (Urinary tract infections (UTI) caused by uropathogenicE. coli) strains in different host genetic background...
YN250422 Macozinone 1377239-83-2
Macozinone (PBTZ169) is a bactericidal benzothiazinone and a potentDprE1(decaprenylphosphoryl-β-d-ribose 2′-oxidase) inhibitor. Macozinone inhibits the essential flavoprotein DprE1 by forming a covalent bond with the active-s...
Ribocil is a highly selective chemical modulator of bacterial riboflavin riboswitches. Ribocil strongly inhibits GFP expression, achieving a 50% effective concentration (EC50) of 0.3μM. in vitro: Ribocil is a highly specific bioac...
SPR719 (VXc-486) is agyrase Binhibitor, with bactericidal activity. SPR719 potently inhibits multiple drug-sensitive isolates and drug-resistant isolates ofMycobacterium tuberculosis, with MICs of 0.03 to 0.30 μg/ml and 0....
YN250489 Sulfadimethoxypyrimidine D4 1392211-88-9
Sulfadimethoxypyrimidine D4 is a deuterium labeled Sulfadimethoxypyrimidine. Sulfadimethoxypyrimidine is a sulfonamide antibiotic with a broad-spectrum antibacterial effect.
YN251360 Tosufloxacin tosylate hydrate 1400591-39-0
Tosufloxacin is a fluoroquinolone antibiotic that is used to treat susceptible infections.
YN250826 ACHN-975 TFA 1410809-37-8
ACHN-975 TFA is a selectiveLpxCinhibitor and exhibits a subnanomolar LpxC inhibitory activity. ACHN-975 TFA is against a wide range of gram-negative bacterias with lowMICvalues (≤1 μg/mL).
YN250304 Zidebactam 1436861-97-0
Zidebactam (WCK-5107) is a potentβ-lactamase inhibitor. Zidebactam also is apenicillin-binding protein2 (PBP2)inhibitor with an IC50 of 0.26 μg/mL.
YN250209 GSK2200150A 1443138-53-1
GSK2200150A, identified by high-throughput screening (HTS) campaign, is an anti-tuberculosis (TB) agent.
Divin, a potent chelator of iron, is a potent inhibitor ofbacterial cell divisionwith bacteriostatic effect inGram-negative and Gram-positive bacteria. Divin disrupts the assembly of late division proteins, reduces peptidoglycan remodel...
TELL : +86-020-82000279
Add:Room 519, Block F, Guangzhou International Business Incubator, No.3 Lanyue Road, Science Town, Huangpu District, Guangzhou, China.
