YN322037 Bunaprolast 99107-52-5

Bunaprolast (U66858) is a potent inhibitor ofLTB4production in human whole blood. Bunaprolast (U66858) also exhibits significant inhibition oflipoxygenase and TXB2release.

YN320254 Proglumide sodium 99247-33-3

Proglumide sodium is a nonpeptide and orally activecholecystokinin (CCK)-A/B receptorsantagonist. Proglumide sodium selective blocksCCK’s effects in the central nervous system (CNS). Proglumide sodium has ability to inhibit...

YN321686 Levodropropizine 99291-25-5

Levodropropizine possess anti-allergic and inhibits histamine receptor, reduces cough by interfering with stimulus activation of peripheral endings of sensory nerves and by modulation of neuropeptides involved in the cough reflex.

YN321304 Rotigotine 99755-59-6

Rotigotine is a dopamine receptor agonist, used in the treatment of Parkinson's disease and restless legs syndrome.

YN321526 Pemirolast potassium 100299-08-9

Pemirolast potassium (BMY 26517) is a histamine H1 antagonist and mast cell stabilizer that acts as an antiallergic agent.

YN290139 Ceramides Mixture 100403-19-8

Ceramides Mixture is an endogenous ceramide and consists of hydroxy and non-hydroxy fatty acid-containing ceramides. Ceramides Mixture is a main lipid component of the permeability barrier in epidermis. Ceramides Mixture is involv...

YN321527 Desloratadine 100643-71-8

Desloratadine is a potent antagonist for human histamine H1 receptor with IC50 of 51 nM.

YN483973 Gastrin I (1-14), human 100940-57-6

Gastrin I (1-14), human is 1-14 fragment of human gastrin I peptide. Gastrin I is an endogenous, gastrointestinal peptide hormone. Gastrin is the major hormonal regulator of gastric acid secretion.

YN321000 Ebrotidine 100981-43-9

Ebrotidine(FI 3542) is a competitive H2-receptor antagonist (Ki= 127.5nM) with a potent antisecretory activity and evidenced gastroprotection.

YN321202 CP-66948 101189-47-3

CP-66948 is ahistamine H2-receptorantagonist with gastric antisecretory activity and mucosal protective properties.

YN322009 Quinotolast sodium 101193-62-8

Quinotolast sodium in the concentration range of 1-100 μg/mL inhibitshistamine,LTC4 and PGD2release in a concentration-dependent manner.

YN321820 Neurokinin B TFA 101536-55-4

Neurokinin B TFA belongs to the tachykinin family of peptides. Neurokinin B binds a family of GPCRs-including neurokinin receptor 1 (NK1R), NK2R, and NK3R-to mediate their biological effect.

YN320973 (Rac)-Rotigotine hydrochlori... 102120-99-0

(Rac)-Rotigotine hydrochloride is a racemate of Rotigotine. Rotigotine is a full agonist ofdopamine receptor, a partial agonist of the5-HT1A receptor, and an antagonist of theα2B-adrenergic receptor, with Kis of 0.71 nM, 4-15 ...

YN321884 Kinetensin 103131-69-7

Kinetensin is aneurotensin-like peptide isolated from pepsin-treated human plasma.

YN481836 Taltirelin 103300-74-9

Taltirelin (TA0910) is a superagonist atthyrotropin-releasing hormone receptor (TRH-R)with an IC50 of 910nM and EC50of 36nM for stimulating an increase in cytosolic Ca2+concentration (Ca2+release).

YN373255 Mirificin 103654-50-8

Mirificin (Puerarin apioside) is a isoflavone inPuerariae LobataeRadix. Mirificin inhibitstyrosinase (TYR)with an IC50 of 12.66μM.

YN320585 Atipamezole 104054-27-5

Atipamezole is a synthetic α2 adrenergic receptor antagonist. It has also been researched in humans as a potential anti-Parkinsonian drug.

YN320584 Atipamezole hydrochloride 104075-48-1

Atipamezole is a synthetic α2 adrenergic receptor antagonist. It has also been researched in humans as a potential anti-Parkinsonian drug. Atipamezole hydrochloride is hydrochloride form of atipamezole.

YN321385 (±)-Bisoprolol hemifumarate 104344-23-2

Bisoprolol fumarate is a selective type β1 adrenergic receptor blocker.

YN321420 Tranilast sodium 104931-56-8

Tranilast sodium (MK-341 sodium) acts as an anti-atopic agent. Tranilast suppresses production ofprostagl and in D2(PGD2,IC50= 0.1 mM). Tranilast sodium exhibits anti-inflammatory and immunomodulatory effects. Tranilast sodiu...