YN321340 Doxylamine succinate 562-10-7

Doxylamine succinate competitively inhibits histamine at H1 receptors with substantial sedative and anticholinergic effects.

YN320449 N-Acetylhistamine 673-49-4

N-Acetylhistamine is a histamine metabolite. N-acetylhistamine can be used as a potential biomarker of histidine metabolism for anaphylactoid reactions.

YN321515 Brompheniramine maleate 980-71-2

Brompheniramine ((±)-Brompheniramine) maleate is a potent and orally active antihistamine of the propylamine class. Brompheniramine maleate is a selectivehistamine H1 receptorantagonist with aKdof 6.06nM. Brompheniramine maleate h...

YN321267 Clemizole hydrochloride 1163-36-6

Clemizole hydrochloride is anH1 histamine receptorantagonist, is found to substantially inhibitHCVreplication. TheIC50 of Clemizole for RNA binding byNS4Bis 24±1nM, whereas itsEC50 for viral replication is 8 µM.

YN321679 Thiethylperazine dimaleate 1179-69-7

Thiethylperazine dimaleate is a phenothiazine derivate, and an orally activedopamine D2-receptor and histamine H1-receptorantagonist. Thiethylperazine dimaleate is also a slectiveABCC1activator that reduces amyloid-β (Aβ) load ...

YN321563 Doxepin Hydrochloride 1229-29-4

Doxepin is a tricyclic antidepressant formulated as a mixture of E-(trans) and Z-(cis) stereoisomers. It inhibits CYP2D6 activity in vivo.

YN321530 Hydroxyzine dihydrochloride 2192-20-3

Hydroxyzine is a histamine H1-receptor antagonist, inhibits binding of [3H]pyrilamine/[3H]desloratadine to human histamine H1 receptor with IC50 of 10 nM/19 nM.

YN321604 Dexchlorpheniramine maleate 2438-32-6

Dexchlorpheniramine maleate is an antihistamine, with anticholinergic properties, used to treat allergic conditions.

YN321605 Antazoline hydrochloride 2508-72-7

Antazoline hydrochloride is a 1st generation antihistamine with also anticholinergic properties used to relieve nasal congestion and in eye drops.

YN321668 Carbinoxamine maleate salt 3505-38-2

Carbinoxamine maleate is a histamine-H1 receptor blocking agent with antihistamine and anticholinergic properties.

YN320780 Oxomemazine 3689-50-7

Oxomemazine is a phenothiazine-basedhistamine H1-receptorblocker with pronounced antimuscarinic properties. Oxomemazine is a selective antagonist formuscarinic M1 receptor, displays about 20-fold difference in the affinity for high (Ki...

YN321164 Decloxizine 3733-63-9

Decloxizine(UCB-1402; NSC289116) is a histamine 1 receptor antagonist.

YN321406 Azatadine 3964-81-6

Azatadine is an histamine and cholinergic inhibitor with IC50 of 6.5nM and 10nM, respectively. Azatadine, a new antihistamine, was evaluated for its efficacy in 20 patients with chronic allergic rhinitis. Eighty percent of patien...

YN321407 Azatadine dimaleate 3978-86-7

Azatadine is an histamine and cholinergic inhibitor with IC50 of 6.5 nM and 10 nM, respectively.

YN320323 Betahistine EP Impurity C 5452-87-9

Betahistine EP Impurity C (NSC19005) is an impurity of Betahistine. Betahistine is a potent, orally active and well-tolerated histamine H1 receptor agonist and H3 receptor antagonist used for the study of rheumatoid arthriti...

YN321523 Betahistine dihydrochloride 5579-84-0

Betahistine is a histamine H3 receptor inhibitor with IC50 of 1.9 μM.

YN321522 Betahistine 5638-76-6

Betahistine Dihydrochloride is a histamine H3 receptors inhibitor used as an antivertigo drug.

YN321759 Nimbin 5945-86-8

Nimbin is a intermediate limonoid isolated fromAzadirachta. Nimbin preventstauaggregation and increases cell viability. Nimbin is effective inhibits theenvelope protein of dengue virus. Nimbin has anti-inflammatory, antipyretic, anti...

YN321640 Triprolidine hydrochloride mo... 6138-79-0

Triprolidine Hydrochloride is the hydrochloride salt form of Triprolidine, which is the first generation histamine H1 antagonist used in allergic rhinitis.

YN321641 Mebhydrolin napadisylate 6153-33-9

Mebhydrolin Napadisylate is classified as an antihistamine drug classes used to treat allergies.