YN321003 Zaltidine 85604-00-8

Zaltidine(CP-57361) is a H2-receptor antagonist, which has the antisecretory action.

YN320361 Emedastine 87233-61-2

Emedastine is a potent, high affinity histamine H1-receptor-selective antagonist with Ki of 1.3 ±0.1 nM for H1-receptors while considerably weaker at H2- (K1 = 49,067 ± 11,113 nM) and H3-receptors (Ki = 12,430 ± 1,282 nM).

YN321696 Emedastine difumarate 87233-62-3

Emedastine Difumarate is the difumarate salt form of emedastine, a second generation, selective histamine H1 receptor antagonist with anti-allergic activity.

YN321660 Acrivastine 87848-99-5

Acrivastine is an antihistamine medicine that relieves the symptoms of allergies.

YN320548 Carebastine 90729-42-3

Carebastine is the active metabolite of Ebastine. Carebastine is ahistamine H1 receptorantagonist. Carebastine inhibits VEGF-induced HUVEC and HPAEC proliferation, migration and angiogenesis in a dose-dependent manner...

YN321559 Ebastine 90729-43-4

Ebastine(LAS-W 090;RP64305) is a long-acting and selective H1-histamine receptor antagonist.

YN320194 Rocastine 91833-49-7

Rocastine is a selective, nonsedatingH1antagonist, acting as an antihistamine.

YN321448 Roxatidine Acetate Hydrochl... 93793-83-0

Roxatidine Acetate Hydrochloride (HOE 760) is a selectivehistamine H2receptorantagonist, can be used for the research of gastric and duodenal ulcers. Roxatidine Acetate Hydrochloride can be rapidly converted to its active metabo...

YN321686 Levodropropizine 99291-25-5

Levodropropizine (DF-526) is a histamine receptor inhibitor, Levodropropizine is an effective and very well tolerated peripheral antitussive drug.

YN321526 Pemirolast potassium 100299-08-9

Pemirolast potassium (BMY 26517) is a histamine H1 antagonist and mast cell stabilizer that acts as an antiallergic agent.

YN321527 Desloratadine 100643-71-8

Desloratadine is a potent antagonist for human histamine H1 receptor with IC50 of 51 nM.

YN321000 Ebrotidine 100981-43-9

Ebrotidine(FI 3542) is a competitive H2-receptor antagonist (Ki= 127.5nM) with a potent antisecretory activity and evidenced gastroprotection.

YN321202 CP-66948 101189-47-3

CP-66948 is ahistamine H2-receptorantagonist with gastric antisecretory activity and mucosal protective properties.

YN322009 Quinotolast sodium 101193-62-8

Quinotolast sodium in the concentration range of 1-100 μg/mL inhibitshistamine,LTC4 and PGD2release in a concentration-dependent manner.

YN322073 CI-949 104961-19-5

CI-949 is an allergic mediator release inhibitor, which inhibitshistamine,leukotriene C4/D4(LTC4/LTD4), and thromboxane B2(TXB2)release with IC50s of 11.4μM, 0.5μM and 0.1μM, respectively.

YN320563 Thioperamide 106243-16-7

Thioperamide (MR-12842) is a potent, orally available, brain penetrant and selectiveH3 receptorantagonist with a Ki of 4.3nM for inhibition of [3H]histamine release. Thioperamide inhibits [3H]histamine synthesis with a Ki of 31n...

YN322050 FRG8701 108498-50-6

FRG-8701 is a newHistamine H2-receptorantagonist with an IC50 of ranging from 0.25 to 0.43μM.

YN321404 Mizolastine 108612-45-9

Mizolastine is a histamine H1-receptor antagonist with IC50 of 47nM used in the treatment of hay fever (seasonal allergic rhinitis), hives and other allergic reactions. Mizolastine is a histamine H1-receptor antagonist with IC50...

YN321549 Epinastine hydrochloride 108929-04-0

Epinastine is an antihistamine and mast cell stabilizer that is used in eye drops to treat allergic conjunctivitis.

YN320201 Wy 49051 113418-56-7

Wy 49051 is a potent, orally activeH1 receptorantagonist, with IC50 of 44nM.