YN370259 EHNA hydrochloride 58337-38-5

EHNA hydrochloride is a potent and selective dual inhibitor ofcyclic nucleotide phosphodiesterase 2 (PDE2)(IC50=4μM) and adenosine deaminase (ADA). EHNA hydrochloride exerts a concentration inhibition of the cGMP-sti...

YN321982 Angiotensin I/II (1-5) 58442-64-1

Angiotensin I/II 1-5 is a peptide that contains the amino acids 1-5, which is converted from Angiotensin I/II. Angiotensin I is formed by the action of renin on angiotensinogen. Angiotensin II is produced from angiotensin I. A...

YN483006 Secoxyloganin 58822-47-2

Secoxyloganin, isolated fromLonicera japonicaThunb, inhibits the blood flow (BF) decrease. Secoxyloganin has allergy-preventive activity.

YN322008 Pamatolol 59110-35-9

Pamatolol is a cardioselectivebeta-adrenoceptorantagonist without sympathomimetic activity.

YN480037 Y-9738 59399-41-6

Y-9738 is a hypolipidemic agent.

YN373336 Glabrol 59870-65-4

Glabrol (Compound 1), One isoprenyl flavonoid was isolated from ethanol extract of licorice roots, is a potent and non-competitiveAcyl-coenzyme A: cholesterol acyltransferase (ACAT)inhibitor with an IC50 value of 24.6μM for r...

YN373332 Vicenin 3 59914-91-9

Vicenin 3 is an angiotensin-converting enzyme (ACE) inhibitor (IC50=46.91μM) from the aerial parts ofDesmodium styracifolium.

YN484228 DU717 59943-31-6

DU-717 is an antihypertensive agent.

YN483025 Oblongine 60008-01-7

Oblongine is isolated from the tuber ofStephania cambodica.

YN321219 Sulprostone 60325-46-4

Sulprostone (SHB 286) is a potent and selectiveEP3 receptoragonist. Sulprostone (SHB 286) is a prostagl and in E2 (PGE2) analogue and has antiulcer and nonsteroidal abortifacient effects. Sulprostone has potential for t...

YN320279 Bufuralol hydrochloride 60398-91-6

Bufuralol hydrochloride (Ro 3-4787 hydrochloride) is a potent non-selective, orally activeβ-adrenoreceptorantagonist with partial agonist activity. Bufuralol hydrochloride is a CYP2D6 probe substrate.

YN360212 P-1075 60559-98-0

P-1075 is a potent activator ofsulfonylurea receptor 2-associated ATP-sensitive potassium channels (SUR2-KIR6), with an EC50 value of 45nM for SUR2B-KIR6 channel activation. P-1075 also P1075 opens mitochondrial K(AT...

YN372901 Amrinone 60719-84-8

Amrinone (Inamrinone) is a positive inotropic-vasodilator agent. Amrinone is a selectivephosphodiesterase IIIinhibitor that increases cyclic adenosine monophosphate by preventing its breakdown. Amrinone is also an orally active, non-...

YN320081 Pirmenol hydrochloride 61477-94-9

Pirmenol hydrochloride inhibits IK.AChby blockingmuscarinic receptors. The IC50 of Pirmenol for inhibition of Carbachol-induced IK.AChis 0.1μM.

YN483910 Fibrinopeptide A, human TF... 61533-47-9

Fibrinopeptide A, human TFA is a 16-residue short polypeptide cleaved from fibrinogen by thrombin. Fibrinopeptide A, human locates at the NH2-termini of the Aα chain.

YN480522 Prolylleucine 61596-47-2

Prolylleucine is a dipeptide containing branched-chain amino acids. Prolylleucine can affect the circadian rhythms and behaviour of animals.

YN481757 Epoprostenol sodium 61849-14-7

Epoprostenol sodium (Prostagl and in I2 (sodium salt)), the synthetic form of the natural prostagl and in derivative prostacyclin (prostagl and in I2), is registered worldwide for the treatment of Pulmonary arterial hypertension (PAH...

YN372785 Captopril 62571-86-2

Captopril is an angiotensin-converting enzyme (ACE) inhibitor with IC50 of 6 nM.

YN482235 Rhodamine 123 62669-70-9

Rhodamine 123 (RH-123, R-22420) is a fluorescent cationic dye used to label mitochondria in living cells. Rhodamine 123 inhibits ADP-stimulated respiration of mitochondria with Ki = 12 μM and ATPase activi...

YN483046 Mulberrin 62949-79-5

Mulberrin is a strong inhibitor of organic anion-transporting polypeptide 2B1 (OATP2B1)-mediated estrone-3-sulfate (E3S) uptake with an IC50 value being 1.8 ±1.5μM.