YN360776 Memantine hydrochloride 41100-52-1

Memantine HCl is a CYP2B6 and CYP2D6 inhibitor for recombinant CYP2B6 and CYP2D6 with Ki of 0.51 nM and 94.9 μM, respectively.

YN321621 Cyproheptadine hydrochloride ... 41354-29-4

Cyproheptadine hydrochloride is non-selective 5HT2 antagonist with IC50 of 0.6 nM. Also a SETD7/9 inhibitor.

YN484356 Pyridoxal 5'-​phosphate mono... 41468-25-1

Pyridoxal 5-phosphate monohydrate is an active vitamin B6 metabolite, which is a cofactor in many reactions of amino acid metabolism.

YN1730017 N6-Cyclopentyladenosine 41552-82-3

N6-Cyclopentyladenosine (CPA) is a selectiveAdenosine A1receptoragonist, with Ki values of 2.3nM, 790nM and 43nM for human A1, A2A and A3receptors, respectively.

YN1730081 A2AR-agonist-1 41552-95-8

A2AR-agonist-1 is a potent A2AR and ENT1 agonist with Ki of 4.39 and 3.47 for A2AR and ENT1. A2AR-agonist-1 is a novel dual-action compound, targeting the Adenosine A2A Receptor and Adenosine Transporter fo...

YN480196 Cresyl Violet perchlorate 41830-80-2

Cresyl Violet perchlorate is a red fluorescent stain, which can be used to stain neurons.

YN321856 D[LEU4,LYS8]-VP 42061-33-6

D[LEU4,LYS8]-VP is a selective agonist ofvasopressin V1breceptor, with theKisof 0.16nM, 0.52nM, and 0.1.38nM for rat, human and mouseV1breceptor, respectively. D[LEU4,LYS8]-VP has weak antidiuretic, vasopressor, ...

YN290077 5-Methoxyflavone 42079-78-7

5-methoxyflavone is a novel DNA polymerase-beta inhibitor and neuroprotective agent against beta-amyloid toxicity.

YN483019 Pinostilbene 42438-89-1

Pinostilbene is a major metabolite of Pterostilbene. Pinostilbene exhibits inhibitory effects on colon cancer cells.

YN482528 Crocin 42553-65-1

Crocin is a water-soluble carotenoid pigment of saffron (Crocus sativus L.). It has been used as a spice for flavoring and coloring food preparations, and in Chinese traditional medicine as an anodyne or tranquilizer.

YN480893 Midodrine 42794-76-3

Midodrine belongs to the class of medications known as vasopressors. It is an adrenergic alpha-1 agonist.

YN320544 Bevantolol hydrochloride 42864-78-8

Bevantolol hydrochloride is a cardioselective, beta adrenoceptor antagonist, devoid of intrinsic β sympathomimetic activity and with weak membrane-stabilizing and local anesthetic properties.

YN360416 Vinpocetine 42971-09-5

Vinpocetine is a selective inhibitor of voltage-sensitive sodium channel for the treatment of stroke, vascular dementia and Alzheimer's disease.

YN480894 Midodrine hydrochloride 43218-56-0

Midodrine hydrochloride is the hydrochloride salt form of midodrine, an adrenergic alpha-1 agonist used as a vasopressor.

YN450078 N-Desmethylnefopam 46868-19-3

N-Desmethylnefopam is the main metabolite of Nefopam. N-Desmethylnefopam is a centrally-acting but non-opioid analgesic agent, for the relief of moderate to severe pain. Nefopam targetsβ-cateninprotein level in mesenchymal cells in-v...

YN373972 (E)-10-Hydroxynortriptyline 47132-16-1

(E)-10-Hydroxynortriptyline (E-10-OH-NT) is a metabolite of Nortriptyline (HY-B1417). Nortriptyline is a tricyclic antidepressant and the main active metabolite of Amitriptyline, and is used to relieve the symptoms of depre...

YN370087 (Z)-10-Hydroxynortriptyline 47132-19-4

(Z)-10-Hydroxynortriptyline is a metabolite of Nortriptyline. Nortriptyline is a tricyclic antidepressant and the main active metabolite of Amitriptyline, and is used to relieve the symptoms of depression.

YN380017 Nitroxazepine 47439-36-1

Nitroxazepine is a tricyclic antidepressant (TCA) for the treatment of depression. Nitroxazepine acts as a serotonin-norepinephrine reuptake inhibitor.

YN321689 Clocapramine 47739-98-0

Clocapramine is an antagonist of theD2,5-HT2Areceptors.

YN380209 Sulindac sulfide 49627-27-2

Sulindac sulfide is a noncompetitiveγ-secretaseinhibitor, with an IC50 of 20.2μM for γ42-secretase activity.