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5-HT Receptor

Chemical structure

Cat.No.

Product Name

CAS no.

Target

  • YN321265 Xanthotoxol 2009-24-7

    Xanthotoxol is a biologically active linear furocoumarin, shows strong pharmacological activities as anti-inflammatory, antioxidant, 5-HT antagonistic, and neuroprotective effects.

  • YN321649 Spiperone hydrochloride 2022-29-9

    Spiperone hydrochloride (Spiroperidol hydrochloride) is a selectivedopamine D2receptor(Kivalues of 0.06nM, 0.6nM, 0.08nM, ~350nM, ~3500nM forD2, D3, D4, D1 and D5receptors, respectively) and 5-HT2A/5-HT1Areceptor(Kis ...

  • YN320055 Flopropione 2295-58-1

    Flopropione is a spasmolytic or antispasmodic agent, and acts as a 5-HT1A receptor antagonist.

  • YN321611 Naftidrofuryl oxalate 3200-06-4

    Nafronyl oxalate salt is the oxalate salt form of nafronyl, which is a selective antagonist of 5-HT2 receptors and a vasodilator used in the management of peripheral and cerebral vascular disorders.

  • YN320841 Cyamemazine 3546-03-0

    Cyamemazine is a neuroleptic agent that contains the phenothiazine chromophore. Cyamemazine is often used as an anxiolytic. Cyamemazine is a potent5-HT3(Kiof 12nM),5-HT2A(Ki= 1.5nM) and 5-HT2C(Kiof 75nM) receptors antagoni...

  • YN321731 Jatrorrhizine 3621-38-3

    Jatrorrhizine, one of the active constituents of Coptis chinensis Franch, has multiple bioactivities, such as hypoglycemic, antimicrobial, and antioxidant activities. It is an inhibitor of AChE with IC50 of 872 nM and demonstrates...

  • YN321711 Puerarin 3681-99-0

    Puerarin (Kakonein), an isoflavones found in the root of Radix puerariae, is a 5-HT2C receptor and benzodiazepine site antagonist.

  • YN320782 5-HT1A modulator 2 hydrochl... 3880-76-0

    5-HT1A modulator 2 hydrochloride, a derivative of 8-OH-DPAT (HY-112061), is a modulator of5-HT1Awith a Ki of 53nM for 5-HT1Abinding.

  • YN321764 Isopteropodine 5171-37-9

    Isopteropodine is heteroyohimbine-type oxindole alkaloid components ofUncaria tomentosa(Willd.) DC. Isopteropodine acts as positive modulators ofmuscarinic M1 and 5-HT2receptors.

  • YN321392 Pizotifen malate 5189-11-7

    Pizotifen Malate is a benzocycloheptane based agent used for recurrent migraine headaches.

  • YN321520 Alverine citrate 5560-59-8

    Alverine citrate is a drug used for functional gastrointestinal disorders.

  • YN320588 Iprindole 5560-72-5

    Iprindole, a tricyclic indole antidepressant, is a weak inhibitor of the uptake of noradrenaline and 5-HT.

  • YN321556 Dihydroergotamine mesylate 6190-39-2

    Dihydroergotamine Mesylate is an ergot derivative with agonistic activity for alpha-adrenergic, serotonergic, and dopaminergic receptors.

  • YN321569 Cyclobenzaprine hydrochloride 6202-23-9

    Cyclobenzaprine HCl is a muscle relaxant by blocking pain sensations, used for the treatment of muscle spasms A 5-HT2 receptor antagonist.

  • YN321730 Jatrorrhizine chloride 6681-15-8

    Jatrorrhizine hydrochloride can inhibit the proliferation and neovascularization of C8161 metastatic melanoma cells with low toxicity, suggests that jatrorrhizine hydrochloride is a potential new antimelanoma drug candidate. Jatrorrhizin...

  • YN321778 Asimilobine 6871-21-2

    Asimilobine is an aporphine isoquinoline alkaloid isolated from plant species ofMagnolia obobataThun. Asimilobine is adopaminebiosynthesis inhibitor and aserotonergic receptorantagonist. Asimilobine shows anantimalarial and anti-can...

  • YN320463 cis-Urocanic acid 7699-35-6

    cis-Urocanic acid is a5-HT2A receptoragonist. cis-Urocanic acid binds to5-HT receptor with relatively high affinity (Kd=4.6nM). cis-Urocanic acid is an immune modulator that induces immunosuppression by binding to the 5-HT2A re...

  • YN321586 Bromperidol 10457-90-6

    Bromperidol is a butyrophenone derivative, is a potent and long-acting neuroleptic, used as an antipsychotic in the treatment of schizophrenia.

  • YN320355 Melitracen hydrochloride 10563-70-9

    Melitracen hydrochloride is a potential dopamine D1/2 receptor antagonist which has antidepressant properties.

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