YN360611 (R)-Baclofen hydrochloride 63701-55-3

(R)-Baclofen hydrochloride (STX 209 hydrochloride) is a selectiveGABAB receptoragonist.

YN420282 Artemisinin 63968-64-9

Artemisinin is a sesquiterpene endoperoxide which is a potent antimalarial agent.

YN321823 Kassinin 63968-82-1

Kassinin is a peptide derived from the Kassina frog. It belongs to tachykinin family of neuropeptides. It is secreted as a defense response, and is involved in neuropeptide signalling.

YN482022 Dipivefrin hydrochloride 64019-93-8

Dipivefrin (Dipivefrine, Propine, Pivalephrine) is a prodrug of epinephrine which is hydrolyzed to epinephrine after absorption into the eye.

YN361065 CGP11952 64078-09-7

CGP11952 is a triazolyl-Benzaphenon resembling the benzodiazepines in its pharmacological action. CGP11952 is an experimentalbenzodiazepinederivative.

YN372312 4'-Hydroxy diclofenac 64118-84-9

4'-Hydroxy diclofenac is an orally active metabolite of Diclofenac (HY-15036) by cytochrome P450 2C9 (CYP2C9). 4'-Hydroxy diclofenac has anti-inflammatory and analgesic properties.

YN361025 Phe-Met-Arg-Phe, amide 64190-70-1

Phe-Met-Arg-Phe, amide dose dependently (ED50=23nM) activates a K+current in the peptidergic caudodorsal neurons.

YN360764 Atracurium besylate 64228-81-5

Atracurium Besylate is a neuromuscular blocking agent with ED95 of 0.2 mg/kg.

YN1730112 Shanzhiside methyl ester 64421-28-9

Shanzhiside methy lester is isolated fromL. rotata. Shanzhiside methyl ester is a small moleculeglucagon-like peptide-1 (GLP-1) receptoragonist and has the ability to induce anti-allodynic tolerance.

YN321418 Tizanidine hydrochloride 64461-82-1

Tizanidine HCl is an α2-adrenergic receptor agonist and inhibits neurotransmitter release from CNS noradrenergic neurons.

YN373203 Glycoursodeoxycholic acid 64480-66-6

Glycoursodeoxycholic acid, a acyl glycine and a bile acid-glycine conjugate, is a metabolite of ursodeoxycholic acid.In Vitro:The antioxidant compound glycoursodeoxycholic acid (GUDCA) fully abrogates UCB-induced cytochrome c ...

YN360121 THIP 64603-91-4

THIP (Gaboxadol) is a selective δ-aminobutyric acid type A receptor (δ-GABAAR) agonist, functionally selective GABAAR lig and , exhibits agonism at α4β1δ, α4β3δ and weak antagonism at αβγ and α4β2δ GAB...

YN483759 Glucagon (19-29), human 64790-15-4

Glucagon (19-29), human is a potent and efficient inhibitor of insulin secretion.

YN380072 MAO-IN-M30 dihydrochlori... 64821-19-8

MAO-IN-M30 dihydrochloride is an orally active, brain-permeable, and brain selective irreversibleMAO-A(IC50=37nM) and MAO-B(IC50=57nM) inhibitor. MAO-IN-M30 dihydrochloride is a potentiron chelator and radical s...

YN480958 Eperisone 64840-90-0

Eperisone is an antispastic agent used for treatment of diseases characterized by muscle stiffness and pain. It works by relaxing both skeletal muscles and vascularsmooth muscles, thus demonstrating avariety of effects such as reducti...

YN370455 Pifithrin-μ 64984-31-2

Pifithrin-μ is a specific p53 inhibitor by reducing its affinity to Bcl-xL and Bcl-2, and also inhibits HSP70 function and autophagy.

YN360421 12,14-Dichlorodehydroabietic ... 65281-77-8

12,14-Dichlorodehydroabietic acid, a chlorinated resin acid, is a potentCa2+-activated K+(BK) channelopener. 12,14-Dichlorodehydroabietic acid blocksGABA-dependent chloride entry in mammalian brain and operates as a non-competi...

YN480546 MS21570 65373-29-7

MS21570 is a selectiveGPR171antagonist, with an IC50 of 220nM.

YN320112 Asenapine 65576-45-6

Asenapine is an antagonist ofserotonin receptors(5-HT2A, 5-HT2B, 5-HT2C, 5-HT6, 5-HT7),adrenoceptors(α1, α2A, α2B, α2C),dopamine receptors(D2, D3, D4) and histamine receptors(H1, H2), withpKis of 8.4-10.5, 8.9-9....

YN484047 Mast cell degranulating pepti... 65636-54-6

Mast cell degranulating peptide (28-49) is a depolarizing agent from bee venom, it can raise the content ofcGMPlevel in mouse cerebellar slices.