YN371053 Glycerophosphoric acid disodi... 154804-51-0

Glycerophosphoric acid disodium salt hydrate is an endogenous metabolite.

YN483960 Calcitonin (8-32), salmon 155069-90-2

Calcitonin (8-32), salmon is a highly selectiveamylin receptorantagonist.

YN360493 Rosiglitazone maleate 155141-29-0

Rosiglitazone, a member of the thiazolidinedione class of antihyperglycaemic agents, is a high-affinity selective agonist of the peroxisome proliferator-activated receptor-γ with IC50 of 42 nM.

YN321699 Mebeverine metabolite O-desm... 155172-67-1

Mebeverine metabolite O-desmethyl Mebeverine alcohol is a metabolite of Mebeverine, which is a potentα1 repectorinhibitor, causing relaxation of the gastrointestinal tract.

YN481540 NB-598 Maleate 155294-62-5

NB-598 Maleate is a potent and competitive inhibitor ofsqualene epoxidase (SE), and suppresses triglyceride biosynthesis through the farnesol pathway.

YN320667 CCK-B Receptor Antagonis... 155412-88-7

CCK-B Receptor Antagonist 2, compound 15b, is a potent and orally activeGastrin/CCK-Bantagonist with an IC50 value of 0.43nM. CCK-B Receptor Antagonist 2 also inhibits gastrin/CCK-A activity with an IC50 of 1.82...

YN320919 Sograzepide 155488-25-8

Sograzepide (Netazepide; YF 476; YM-220) is an extremely potent , highly selective  and orally activeGastrin/CCK-Bantagonist with an IC50 value of 0.1nM, has inhibitory effect on Gastrin/CCK-A activity with an IC5...

YN483483 25-O-Methylalisol A 155801-00-6

25-O-Methylalisol A is a protostane triterpenoids isolated fromAlisma orientale. The dried rhizomes of the aquatic plantAlisma orientaleknown as Rhizoma Alismatis is a common traditional Chinese medicine used for diuretic, anti-inf...

YN320711 Alvimopan 156053-89-3

Alvimopan (LY-246736) is a potent, relatively nonselective opioid antagonist with Ki values of 0.77, 4.4, and 40 nM for the μ, δ, and κ opioid receptors, respectively, displaying >100-fold selectivity over other aminer...

YN480651 BIBB 515 156635-05-1

BIBB 515 is a potent, selective and orally active2,3-oxidosqualene cyclase (OSC)inhibitor withED50values of 0.2-0.5 mg/kg and 0.36-33.3 mg/kg in rats and mice (1-5 hours), respectively. BIBB 515 exerts lipid-lowering effe...

YN481260 N1,N11-Diethylnorspermine t... 156886-85-0

N1,N11-Diethylnorspermine tetrahydrochloride (DENSPM tetrahydrochloride) potently inducesSSAT (spermidine/spermine N1-acetyltransferase)mRNA and effectively stabilizes SSAT enzyme activity.

YN481531 BPH-652 157124-84-0

BPH-652 is aS. aureusdehydrosqualene synthase (CrtM)inhibitor, with a Ki of 1.5nM and an IC50 of 100-300nM (S. aureuspigment formation).

YN482917 Gypenoside A 157752-01-7

Gypenoside A is a natural compound isolaated fromGynostemma pentaphyllum Makino.

YN250581 Rimonabant Hydrochloride 158681-13-1

Rimonabant Hydrochloride (SR 141716A Hydrochloride) is a highly potent and selective centralcannabinoid receptor (CB1)antagonist with an Ki of 1.8nM. Rimonabant hHydrochloride (SR 141716A Hydrochloride) also inhibitsMycob...

YN360981 Bisandrographolide C 160498-02-2

Bis and rographolide C is an unusual dimer of ent-labdane diterpenoid isolated and identified from and rographis paniculata. Bis and rographolide C activatesTRPV1 and TRPV3channels withKdvalues of 289 and 341μM respective...

YN483727 Elcatonin acetate 160649-04-7

Elcatonin (Carbocalcitonin) acetate is a synthetic analog of eel calcitonin. Elcatonin acetate increases bone mineral density, inhibits bone resorption and processes a central analgesic effect.

YN480565 DMG-PEG 2000 160743-62-4

DMG-PEG 2000 is used for the preparation of liposome forsiRNA deliverywith improved transfection efficiency in vitro. DMG-PEG 2000 is also used for the lipid nanoparticle for an oral plasmid DNA delivery approach in vivo...

YN1720036 GLP-1(9-36)amide 161748-29-4

GLP-1(9-36)amide is a major metabolite of glucagon-like peptide-1-(7-36) amide formed by the enzyme dipeptidyl peptidase-4 (DPP-4). GLP-1(9-36)amide acts as an antagonist to the human pancreaticGLP-1 receptor.

YN483720 Pulsatilloside C 162341-28-8

Pulsatilloside C is a phenolic compound isolated fromPulsatilla koreana. Pulsatilloside C significantly inhibits adipocyte differentiation.

YN480051 UK-157147 162704-20-3

UK-157147 is a substrate for UDP-glucuronosyltransferases (UGT1A1) with a Km value of 105μM.