YN321985 β-Endorphin, equine 79495-86-6

β-Endorphin, equine is an endogenous opioid peptide, which binds at high affinity to bothμ/δ opioid receptors. Analgesic properties.

YN380167 Sertraline hydrochloride 79559-97-0

Sertraline HCl is a 5-HT antagonist with Ki of 13 nM.

YN482720 Crassicauline A 79592-91-9

Crassicauline A (Crassicaulin A) is a bioactive alkaloid found in roots ofAconitum carmichaeli. Crassicauline A (Crassicaulin A) possesses feeding deterrent activity againstT. castaneumadults with an EC50of 1134.5 ppm.

YN322007 (±)-Tazifylline 79712-55-3

(±)-Tazifylline is a potent, selective and long-actinghistamine H1 receptorantagonist.

YN320891 Idazoxan hydrochloride 79944-56-2

Idazoxan hydrochloride (RX 781094 hydrochloride) is anα2-adrenoceptorantagonist and is also aimidazoline receptors (IRs)antagonist competitively antagonized the centrally induced hypotensive effect of imidazoline-like drugs (IMs)....

YN321969 Dynorphin A 1-10 79994-24-4

Dynorphin A (1-10) an endogenous opioid neuropeptide, binds to extracellular loop 2 of theκ-opioid receptor. Dynorphin A (1-10) also blocksNMDA-activated current with an IC50 of 42.0μM.

YN482425 Helicid 80154-34-3

Helicide (4-formylphenyl-O-β-d-allopyranoside), a main active constituent from seeds of the Chinese herb Helicia nilagirica, has been reported to exert a sedative, analgesic and hypnotic effect, and is used clinically to treat neurasth...

YN360008 Pipequaline hydrochloride 80221-58-5

Pipequaline hydrochloride (PK-8165 hydrochloride) is a partialbenzodiazepine receptoragonist with anxiolytic activity.

YN370128 AR7 80306-38-3

AR7 is a retinoic acid receptor α (RARα) antagonist.

YN482608 Notoginsenoside R2 80418-25-3

Notoginsenoside R2 is a newly isolated notoginsenoside from Panax notoginseng, showed neuroprotective effects against 6-OHDA-induced oxidative stress and apoptosis.

YN321917 Dynorphin A 80448-90-4

Dynorphin A, an endogenous opioid peptide, is a highy potentkappa opioid receptor (KOR)activator. Dynorphin A also serve as an agonist for other opioid receptors,  such as mu (MOR) and delta (DOR).

YN321718 Sec-O-Glucosylhamaudol 80681-44-3

Sec-O-Glucosylhamaudol is a natural compound extracted fromPeucedanum japonicum Thunb, decreases levels ofμ-opioid receptor, with analgesic effect.

YN484006 β-Casomorphin (1-3), amide 80705-23-3

β-Casomorphin (1-3), amide is a peptide fragment of β-Casomorphin with 3 amino acid.

YN1730020 SKF-82958 80751-65-1

SKF-82958 ((±)-SKF 82958) is adopamine D1 receptorfull agonist (K0.5=4nM), displays selective for D1 over D2 receptors (K0.5=73nM). SKF-82958 induces dopamine D1 receptor-dependent adenylate cyclase activity in rat striat...

YN320823 Cisapride 81098-60-4

Cisapride is a nonselective 5-HT4 receptor agonist with gastroprokinetic effects.

YN1730011 L-741626 81226-60-0

L-741626 is a selectiveD2 dopamine receptorantagonist, with theKivalues of 2.4, 100 and 220nM for human D2, D3 and D4 receptors respectively.

YN483916 Somatostatin-28 1-12 81286-16-0

Somatostatin-28 (1-12) is a somatostatin fragment that is monitored in brain tissue to track processing of somatostatin.

YN1730073 Amisulpride hydrochloride 81342-13-4

Amisulpride hydrochloride is a dopamineD2/D3receptorantagonist with Kis of 2.8 and 3.2nM for hum and opamine D2 and D3, respectively.

YN1730003 Pentiapine 81382-51-6

Pentiapine (CGS 10746) is adopamine releaseinhibitor without binding to synaptic dopamine receptor sites.

YN320199 Spirendolol 81840-58-6

Spirendolol is aβ adrenergic receptorantagonist.