Chemical structure
Cat.No.
Product Name
CAS no.
Target
YN380096 Escitalopram 128196-01-0
Escitalopram ((S)-Citalopram), the S-enantiomer of racemic Citalopram, is a selectiveserotonin reuptakeinhibitor (SSRI) with a Ki of 0.89nM. Escitalopram has ∼30 fold higher binding affinity than its R(-)-enantiomer and show...
YN322088 5-HT3 antagonist 2 128199-93-9
5-HT3 antagonist 2 is a5-HT3receptor antagonist.
YN321868 MCH(human, mouse, rat) 128315-56-0
MCH (human, mouse, rat) is a potent peptide agonist ofMCH-R and exhibits bindingIC50 values of 0.3nM and 1.5nM for MCH1R and MCH2R, respectively. MCH (human, mouse, rat) is a highly sensitive to MCH-2R in a C...
YN480684 Sauristolactam 128533-02-8
Sauristolactam, a natural aristolactam isolated from aerial portions ofSaururus chinensis, has significant neuroprotective activity against glutamate-induced toxicity in primary cultured rat cortical cells. Sauristolactam also inhibits t...
YN1730013 NMI 8739 129024-87-9
NMI 8739 is adopamine D2autoreceptoragonist, which is an amine conjugate of the DHA carrier and the neurotransmitter dopamine.
YN320101 Ocaperidone 129029-23-8
Ocaperidone is an effective antipsychotic agent, acting as a potent5-HT2 and dopamine D2antagonist, and a5-HT1Aagonist, with Kis of 0.14nM, 0.46nM, 0.75nM, 1.6nM and 5.4nM for 5-HT2, a1-adrenergic receptor, dopamine D2, ...
YN380039 Rivastigmine tartrate 129101-54-8
Rivastigmine Tartrate is a cholinesterase inhibitor with IC50 of 5.5 μM, and used as a parasympathomimetic or cholinergic agent for the treatment of mild to moderate Alzheimer disease.
YN321809 Rat CGRP-(8-37) 129121-73-9
Rat CGRP-(8-37) (VTHRLAGLLSRSGGVVKDNFVPTNVGSEAF) is a highly selectiveCGRP receptorantagonist.
YN361078 Gidazepam 129186-29-4
Gidazepam is an agonist ofGABA receptor channels(GABA RCs).
YN380280 Autocamtide 2 129198-88-5
Autocamtide 2 is a highly selective peptide substrate of calcium/calmodulin-dependent protein kinase II (CaMKII). It can be used in the CaMKII activity assay.
YN321567 Perospirone hydrochloride 129273-38-7
Perospirone is an atypical or second-generation antipsychotic of the azapirone family that antagonizes serotonin 5HT2A receptors and dopamine D2 receptors. It also displays affinity towards 5HT1A receptors as a partial agonist.
YN380242 Semilicoisoflavone B 129280-33-7
Semilicoisoflavone B, an isoflavone, mainly derived fromGlycyrrhiza uralensisFisch.. Semilicoisoflavone B reducesamyloid β(Aβ) secretion by inhibiting β-secretase-1 (BACE1) expression and activity. Semilicoisoflavone B dec...
YN322076 5-HT3 antagonist 1 129294-09-3
5-HT3 antagonist 1 is a potent and selective antagonist ofserotonin 3 (5-HT3) receptor.
YN320168 (±)-Fabesetron hydrochloride 129299-81-6
(±)-Fabesetron hydrochloride ((±)-FK1052) is the racemate of Fabesetron hydrochloride, which is a potent5-HT3 and 5-HT4receptor dual antagonist.
YN320281 Fabesetron 129300-27-2
Fabesetron (FK1052) is an orally active5-HT3receptorantagonist with5-HT4receptorantagonistic activity. Fabesetron (FK1052) can be used in the study for both acute and delayed emesis induced by cancer chemotherapy.
GR 82334 is a potent and specific reversibletachykinin NK1 receptorantagonist. GR 82334 inhibits substance P-induced sensitization by blocking SP NK1 receptors in naked mole-rats.
YN440197 Sp-8-CPT-cAMPS 129693-13-6
Sp-8-CPT-cAMPS, a cAMP analog, is a potent and selective activator of the cAMP-dependentprotein kinas A (PKA I and PKA II). Sp-8-CPT-cAMPS selects site A of RI compares to site A of RII by 153-fold...
YN320883 Aripiprazole 129722-12-9
Aripiprazole is a novel atypical antipsychotic drug that is reported to be a high-affinity 5-HT receptor partial agonist.
YN320070 Dehydroaripiprazole 129722-25-4
Dehydroaripiprazole (OPC-14857) is an active metabolite of Aripiprazole. Aripiprazole is an antipsychotic agent and is metabolized by CYP3A4 and CYP2D6 forming mainly Dehydroaripiprazole. Dehydroaripiprazole has with ant...
YN440196 Rp-8-CPT-cAMPS 129735-01-9
Rp-8-CPT-cAMPS, a cAMP analog, is a potent and competitive antagonist of cAMP-induced activation of cAMP-dependentPKA I and II. Rp-8-CPT-cAMPS preferentially selects site A of RI compares to site A of R...
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