YN321061 Rapacuronium bromide 156137-99-4

Rapacuronium bromide is an allosteric modulator of muscarinic acetylcholine receptor (mAChR).

YN360020 SX-3228 156364-04-4

SX-3228 is a selectivebenzodiazepine1(BZ1) receptor agonist with an IC50 of 17nM.

YN1730040 FSCPX 156547-56-7

FSCPX is a potent and selective irreversible antagonist ofA1adenosine receptor (A1AR), with low nanomolar potency for binding to the A1AR. FSCPX could modifies the effect of NBTI, a nucleoside transport inhibitor, by ...

YN330694 S-MTC 156719-41-4

S-MTC is a selective type I nitric oxide synthase (NOS) inhibitor.

YN320111 SNC80 156727-74-1

SNC80 (NIH 10815) is a potent, highly selective and non-peptideδ-opioid receptoragonist with a Ki of 1.78nM and an IC50 of 2.73nM. SNC80 also selectively activatesμ-δ heteromerin HEK293 cells with an EC50 of 52.8nM...

YN360623 Omberacetam 157115-85-0

Omberacetam (GVS-111) is a medication promoted and prescribed in Russia and neighbouring countries as a nootropic.

YN483243 Bacoside A3 157408-08-7

Bacoside A3, a triterpenoid saponin, is one of the major active constituents inBacopa monnieri. Bacoside A3 has neuroprotective activity.

YN360138 (S)-SNAP5114 157604-55-2

(S)-SNAP5114 is a selectiveGABA transportinhibitor, with IC50 values of 5μM and 21μM for hGAT-3 and rGAT-2, respectively. (S)-SNAP5114 is an anticonvulsant drug.

YN361036 ω-Agatoxin TK 158484-42-5

ω-Agatoxin TK, a peptidyl toxin of the venom ofAgelenopsis aperta, is a potent and selectiveP/Q type Ca2+channelblocker. ω-Agatoxin TK inhibits the high K+depolarisation-induced rise in internal Ca2+in cerebral isolated nerv...

YN1730006 (+)-Dihydrexidine hydrochlori... 158704-02-0

(+)-Dihydrexidine hydrochloride ((+)-DAR-0100 hydrochloride) is adopamine D1 receptoragonist with an EC50 of 72± 21nM.

YN320334 GR 159897 158848-32-9

GR 159897 is a highly potent, selective, competitive, brain-penetrated non-peptideneurokinin 2 (NK2) receptorantagonist. GR 159897 has little or no affinity for NK1 and NK3receptors. GR 159897 inhibits binding of [3H]GR10067...

YN321911 GR231118 158859-98-4

GR231118, an analogue of the C-terminus of neuropeptide Y, is a potent , competitive and relative seletive antagonist at humanneuropeptide Y Y receptor with a pKi of 10.4. GR231118 a potent agonist at the human neuropeptide Y Y...

YN321674 Frovatriptan succinate 158930-09-7

Frovatriptan Succinate is the succinate salt form of frovatriptan, a synthetic triptan with serotonin (5-HT) receptor agonist activity especially for the 5-HT1B/1D receptors.

YN321673 Frovatriptan succinate hydrat... 158930-17-7

Frovatriptan succinate hydrate ((R)-Frovatriptan succinate hydrate) is a potent, high affinity, selective and orally active5-HT1B(pK50of 8.2) and 5-HT1Dreceptoragonist. Frovatriptan succinate hydrate exhibits >10-fold selectiv...

YN1730063 L-745870 158985-00-3

L-745870 is a potent, selective, brain-penetrant and orally activedopamine D4receptorantagonist with aKiof 0.43nM. L-745870 shows weaker affinity for D2(Kiof 960nM) and D3(Kiof 2300nM) receptors, and exhibits moderate affin...

YN361026 Phe-Met-Arg-Phe amide trif... 159237-99-7

Phe-Met-Arg-Phe amide trifluoroacetate is an activator of K+current, with ED50of 23nM in the peptidergic caudodorsal neurons.

YN360075 MPDC 159262-32-5

MPDC is a potent and competitive inhibitor of the Na+-dependent high-affinityglutamate transporterin forebrain synaptosomes.

YN484223 SZ1676 159325-23-2

SZ1676 is a derivative of SZ1677, which is a neuromuscular blocking agent.

YN360376 SCH 50911 hydrochloride 160415-07-6

SCH 50911 hydrochloride, (+)-(S)-5,5-dimethylmorpholinyl-2-acetic acid, a selective, orally-active and competitive γ-Aminobutyric acid BGABA(B)receptor antagonist, binds to GABA(B) receptor with IC50 of 1.1μM. SCH ...

YN371583 4-Desmethyl Istradefylline 160434-48-0

4-Desmethyl Istradefylline is a metabolite of Istradefylline. 4-Istradefylline is a very potent, selective and orally activeadenosine A2A receptorantagonist with Kiof 2.2nM in experimental models of Parkinson's disease.