Chemical structure
Cat.No.
Product Name
CAS no.
Target
CFM-2 is a potent and selective non-competitiveAMPARantagonist. CFM-2 possesses anticonvulsant activity in various models of seizures.
YN361017 13-Hydroxyisobakuchiol 178765-49-6
Hydroxyisobakuchiol (Delta3,2-Hydroxylbakuchiol), an analog of Bakuchiol (HY-N0235) isolated fromPsoralea corylifolia(L.), is a potentmonoamine transporterinhibitor. 13-Hydroxyisobakuchiol is more selective for the dopamine transp...
YN360678 UK-240455 178908-09-3
UK-240455 is a potent and selective N-methyl D-aspartate (NMDA) glycine site antagonist.
C-DIM12 is Nurr1 activator that stimulates Nurr1 mediated apoptosis axis in bladder cancer cells and tumors and inhibits NF-κB–dependent gene expression in glial cells.
YN481418 (Z)-MDL 105519 179105-67-0
(Z)-MDL 105519 is the inactive isoform of MDL 105519.
YN1730090 Sumanirole maleate 179386-44-8
Sumanirole maleate (U-95666E; PNU-95666E) is a highly selectiveD2 receptorfull agonist with anED50of about 46nM. Sumanirole was developed for the treatment of Parkinson's disease and restless leg syndrome.
YN360404 SDZ 220-581 hydrochloride 179411-93-9
SDZ 220-581 hydrochloride is an orally active, potent, competitiveNMDA receptorantagonist withpKivalue of 7.7.
YN360403 SDZ 220-581 Ammonium salt 179411-94-0
SDZ 220-581 Ammonium salt is an orally active, potent, competitiveNMDA receptorantagonist withpKivalue of 7.7.
YN320824 Prucalopride 179474-81-8
Prucalopride is a selective, high affinity 5-HT receptor agonist for 5-HT4A and 5-HT4B receptor with Ki of 2.5 nM and 8 nM, respectively, exhibits >290-fold selectivity against other 5-HT receptor subtypes.
YN321258 Eptapirone 179756-58-2
Eptapirone (F11440) is a potent, selective, high efficacy 5-HT1A receptor agonist with marked anxiolytic and antidepressant potential.
YN320102 SB-224289 hydrochloride 180084-26-8
SB-224289 hydrochloride is a selective5-HT1B receptorantagonist, with anxiolytic effect.
YN321118 Tezosentan 180384-57-0
Tezosentan (RO 610612) is anendothelin (ET)receptor antagonist, withpA2sof 9.5, 7.7 for ETA and ETBreceptors, respectively.
YN321702 Solifenacin hydrochloride 180468-39-7
Solifenacin hydrochloride (YM905 hydrochloride) is amuscarinic receptorantagonist, withpKis of 7.6, 6.9 and 8.0 forM1,M2 and M3receptors, respectively.
AF40431, the first reported small-molecule lig and of sortilin, has an IC50 of 4.4 µM and aKdof 0.7 µM . AF40431 is bound in the neurotensin-binding site of sortilin.
YN321477 Almotriptan malate 181183-52-8
Almotriptan Malate is a selective 5-hydroxytryptamine1B/1D (5-HT1B/1D) receptor agonist, used for the treatment of Migraine attacks in adults.
YN380299 β-Amyloid (10-35), amide 181427-66-7
β-Amyloid (10-35), amide is composed of 26 aa (10-35 residues of the Aβ peptide) and is the primary component of the amyloid plaques of Alzheimer’s disease.
SB228357 is a selective, potent and orall active5-HT2C/2Breceptorantagonist with pKi values. of 6.9, 8.0 and 9.0 for5-HT2A,5-HT2B and 5-HT2C, respectively. SB228357 has antidepressant/anxiolytic effects.
YN320732 SB 242084 181632-25-7
SB 242084 is a 5-HT2C receptor antagonist(pKi=9.0) that displays 158- and 100-fold selectivity over 5-HT2A and 5-HT2B receptors respectively.
DPI-3290 (Org 41793) is a potent and specificopioid receptorsagonist with Ki values of 0.18nM, 0.46nM, and 0.62nM for δ-, μ-, and κ-opioid receptors, respectively。DPI-3290 is one of a series of novel centrally acting ag...
LY334370 is a selective5-HT1Freceptor agonist with a Ki of 1.6nM.
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